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Chemmedchem|January 16, 2018
Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside MacrophagesMarco Paolino, Margherita Brindisi, Alessandra Vallone, et al.European Journal of Medicinal Chemistry|September 14, 2019
Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systemsAlessandro Grillo, Giulia Chemi, Simone Brogi, et al.Journal of Medicinal Chemistry|February 16, 2011
Non-nucleoside inhibitors of human adenosine kinase: synthesis, molecular modeling, and biological studiesStefania Butini, Sandra Gemma, Margherita Brindisi, et al.ACS Chemical Neuroscience|April 23, 2021
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic AgentsAlessandro Grillo, Filomena Fezza, Giulia Chemi, et al.Journal of Medicinal Chemistry|November 14, 2012
Mimicking the intramolecular hydrogen bond: synthesis, biological evaluation, and molecular modeling of benzoxazines and quinazolines as potential antimalarial agentsSandra Gemma, Caterina Camodeca, Margherita Brindisi, et al.European Journal of Medicinal Chemistry|May 7, 2016
Development of novel cyclic peptides as pro-apoptotic agentsMargherita Brindisi, Samuele Maramai, Simone Brogi, et al.Journal of Medicinal Chemistry|February 19, 2016
Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and PainMargherita Brindisi, Samuele Maramai, Sandra Gemma, et al.Journal of Medicinal Chemistry|July 13, 2012
Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profilingSandra Gemma, Caterina Camodeca, Salvatore Sanna Coccone, et al.Journal of Medicinal Chemistry|January 19, 2024
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological CharacterizationStefania Butini, Uwe Grether, Kwang-Mook Jung, et al.European Journal of Medicinal Chemistry|May 13, 2022
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viabilityStefano Federico, Tuhina Khan, Anna Fontana, et al.Pageof 9