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Stefano Pieraccini

Showing results (41-50 of 55) with videos related to

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European Journal of Medicinal Chemistry|April 30, 2016
4-(1,2-diarylbut-1-en-1-yl)isobutyranilide derivatives as inhibitors of topoisomerase IIMichael S Christodoulou, Mikel Zarate, Francesca Ricci, et al.
Organic & Biomolecular Chemistry|April 20, 2023
Synthesis of SARS-CoV-2 M<sup>pro</sup> inhibitors bearing a cinnamic ester warhead with <i>in vitro</i> activity against human coronavirusesAndrea Citarella, Davide Moi, Martina Pedrini, et al.
Bioorganic & Medicinal Chemistry|November 7, 2024
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cellsAndrea Citarella, Serena Petrella, Davide Moi, et al.
Chemmedchem|October 23, 2012
Camptothecin-7-yl-methanthiole: semisynthesis and biological evaluationMichael S Christodoulou, Franco Zunino, Valentina Zuco, et al.
Bioorganic & Medicinal Chemistry|May 28, 2025
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 M<sup>pro</sup> and cathepsins for broad-spectrum anti-coronavirus activityAndrea Citarella, Giulia Sibille, Davide Moi, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|November 17, 2021
Maytansinol Derivatives: Side Reactions as a Chance for New Tubulin BindersPaola Marzullo, Zlata Boiarska, Helena Pérez-Peña, et al.
Bioorganic & Medicinal Chemistry|February 25, 2025
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocksMartina Pedrini, Luca Pozzi, Francesca Sacchi, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|January 24, 2023
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule DynamicsZlata Boiarska, Helena Pérez-Peña, Anne-Catherine Abel, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|December 5, 2022
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule DynamicsZlata Boiarska, Helena Pérez-Peña, Anne-Catherine Abel, et al.
ACS Medicinal Chemistry Letters|April 20, 2018
Imidazo[2,1-<i>b</i>]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid ReceptorMichael S Christodoulou, Federico Dapiaggi, Francesca Ghiringhelli, et al.
Pageof 6

Showing results (41-50 of 55) with videos related to

Sort By:
Pageof 6
European Journal of Medicinal Chemistry|April 30, 2016
4-(1,2-diarylbut-1-en-1-yl)isobutyranilide derivatives as inhibitors of topoisomerase IIMichael S Christodoulou, Mikel Zarate, Francesca Ricci, et al.
Organic & Biomolecular Chemistry|April 20, 2023
Synthesis of SARS-CoV-2 M<sup>pro</sup> inhibitors bearing a cinnamic ester warhead with <i>in vitro</i> activity against human coronavirusesAndrea Citarella, Davide Moi, Martina Pedrini, et al.
Bioorganic & Medicinal Chemistry|November 7, 2024
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cellsAndrea Citarella, Serena Petrella, Davide Moi, et al.
Chemmedchem|October 23, 2012
Camptothecin-7-yl-methanthiole: semisynthesis and biological evaluationMichael S Christodoulou, Franco Zunino, Valentina Zuco, et al.
Bioorganic & Medicinal Chemistry|May 28, 2025
Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 M<sup>pro</sup> and cathepsins for broad-spectrum anti-coronavirus activityAndrea Citarella, Giulia Sibille, Davide Moi, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|November 17, 2021
Maytansinol Derivatives: Side Reactions as a Chance for New Tubulin BindersPaola Marzullo, Zlata Boiarska, Helena Pérez-Peña, et al.
Bioorganic & Medicinal Chemistry|February 25, 2025
Design, synthesis and in vitro validation of bivalent binders of SARS-CoV-2 spike protein: Obeticholic, betulinic and glycyrrhetinic acids as building blocksMartina Pedrini, Luca Pozzi, Francesca Sacchi, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|January 24, 2023
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule DynamicsZlata Boiarska, Helena Pérez-Peña, Anne-Catherine Abel, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|December 5, 2022
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule DynamicsZlata Boiarska, Helena Pérez-Peña, Anne-Catherine Abel, et al.
ACS Medicinal Chemistry Letters|April 20, 2018
Imidazo[2,1-<i>b</i>]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid ReceptorMichael S Christodoulou, Federico Dapiaggi, Francesca Ghiringhelli, et al.
Pageof 6