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Journal of Biomolecular Screening|August 16, 2013
Are GPCRs still a source of new targets?Stephen L GarlandCurrent Topics in Medicinal Chemistry|April 8, 2011
A ligand's view of target similarity: chemogenomic binding site-directed techniques for drug discoveryStephen L Garland, David E GloriamJournal of Medicinal Chemistry|June 23, 2009
Definition of the G protein-coupled receptor transmembrane bundle binding pocket and calculation of receptor similarities for drug designDavid E Gloriam, Steven M Foord, Frank E Blaney, et al.Biochemical and Biophysical Research Communications|November 17, 2009
Non-peptidic antagonists of the CGRP receptor, BIBN4096BS and MK-0974, interact with the calcitonin receptor-like receptor via methionine-42 and RAMP1 via tryptophan-74Philip S Miller, James Barwell, David R Poyner, et al.Chemical Science|August 30, 2018
The creation and characterisation of a National Compound Collection: the Royal Society of Chemistry pilotDavid M Andrews, Laura M Broad, Paul J Edwards, et al.Bioorganic & Medicinal Chemistry Letters|April 18, 2003
5-aryl-pyrazolo[3,4-b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3)Jason Witherington, Vincent Bordas, Stephen L Garland, et al.Journal of Medicinal Chemistry|January 17, 2009
The discovery of a selective, small molecule agonist for the MAS-related gene X1 receptorBerthold Wroblowski, Mark J Wigglesworth, Philip G Szekeres, et al.Bioorganic & Medicinal Chemistry Letters|December 17, 2009
The identification of structurally novel, selective, orally bioavailable positive modulators of mGluR2Pier L D'Alessandro, Corrado Corti, Adelheid Roth, et al.Bioorganic & Medicinal Chemistry Letters|January 26, 2010
Potent oxadiazole CGRP receptor antagonists for the potential treatment of migrainePaula L Nichols, Jonathan Brand, Michael Briggs, et al.Pageof 1