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Chemistry & Biology|November 2, 2010
Structural determinants of inhibitor selectivity in prokaryotic IMP dehydrogenasesDeviprasad R Gollapalli, Iain S Macpherson, George Liechti, et al.Journal of Medicinal Chemistry|September 3, 2010
Amino derivatives of indole as potent inhibitors of isoprenylcysteine carboxyl methyltransferaseMei-Lin Go, Jo Lene Leow, Suresh Kumar Gorla, et al.Acta Crystallographica. Section F, Structural Biology Communications|May 7, 2015
Structure of Cryptosporidium IMP dehydrogenase bound to an inhibitor with in vivo antiparasitic activityYoungchang Kim, Magdalena Makowska-Grzyska, Suresh Kumar Gorla, et al.Journal of Medicinal Chemistry|September 7, 2012
Selective and potent urea inhibitors of cryptosporidium parvum inosine 5'-monophosphate dehydrogenaseSuresh Kumar Gorla, Mandapati Kavitha, Minjia Zhang, et al.Journal of the American Chemical Society|January 8, 2010
The structural basis of Cryptosporidium -specific IMP dehydrogenase inhibitor selectivityIain S Macpherson, Sivapriya Kirubakaran, Suresh Kumar Gorla, et al.Bioorganic & Medicinal Chemistry Letters|January 18, 2013
Phthalazinone inhibitors of inosine-5'-monophosphate dehydrogenase from Cryptosporidium parvumCorey R Johnson, Suresh Kumar Gorla, Mandapati Kavitha, et al.Bioorganic & Medicinal Chemistry Letters|February 8, 2012
Structure-activity relationship study of selective benzimidazole-based inhibitors of Cryptosporidium parvum IMPDHSivapriya Kirubakaran, Suresh Kumar Gorla, Lisa Sharling, et al.The Journal of Biological Chemistry|January 10, 2015
A novel cofactor-binding mode in bacterial IMP dehydrogenases explains inhibitor selectivityMagdalena Makowska-Grzyska, Youngchang Kim, Natalia Maltseva, et al.Antimicrobial Agents and Chemotherapy|December 25, 2013
Validation of IMP dehydrogenase inhibitors in a mouse model of cryptosporidiosisSuresh Kumar Gorla, Nina N McNair, Guangyi Yang, et al.Journal of Medicinal Chemistry|May 15, 2013
Optimization of benzoxazole-based inhibitors of Cryptosporidium parvum inosine 5'-monophosphate dehydrogenaseSuresh Kumar Gorla, Mandapati Kavitha, Minjia Zhang, et al.Pageof 2