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Frontiers in Neuroscience|January 1, 2021
Anti-sortilin1 Antibody Up-Regulates Progranulin via Sortilin1 Down-RegulationShuuichi Miyakawa, Hiroyuki Sakuma, Dnyaneshwar Warude, et al.Bioorganic & Medicinal Chemistry|April 28, 2016
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel non-basic 1-(2H-indazole-5-yl)pyridin-2(1H)-one derivatives and mitigation of mutagenicity in Ames testHideyuki Igawa, Masashi Takahashi, Minoru Ikoma, et al.The Journal of Pharmacology and Experimental Therapeutics|October 23, 2022
Quantitative Model Analysis and Simulation of Pharmacokinetics and Metastasis-Associated Lung Adenocarcinoma 1 RNA Knockdown Effect After Systemic Administration of Cholesterol-Conjugated DNA/RNA Heteroduplex Oligonucleotide Crossing Blood-Brain Barrier of MiceAkihiko Goto, Syunsuke Yamamoto, Tomoko Igari, et al.Journal of Medicinal Chemistry|January 7, 2016
Melanin-Concentrating Hormone Receptor 1 Antagonists Lacking an Aliphatic Amine: Synthesis and Structure-Activity Relationships of Novel 1-(Imidazo[1,2-a]pyridin-6-yl)pyridin-2(1H)-one DerivativesHideyuki Igawa, Masashi Takahashi, Keiko Kakegawa, et al.Nature Communications|September 26, 2024
Heteroduplex oligonucleotide technology boosts oligonucleotide splice switching activity of morpholino oligomers in a Duchenne muscular dystrophy mouse modelJuri Hasegawa, Tetsuya Nagata, Kensuke Ihara, et al.The Journal of Pharmacology and Experimental Therapeutics|February 17, 2026
Preclinical characterization of pharmacokinetics, enzyme occupancy, and pharmacodynamics of soticlestat (TAK-935), a novel cholesterol 24-hydroxylase inhibitorMaki Miyamoto, Toshiya Nishi, Tatsuki Koike, et al.Bioorganic & Medicinal Chemistry|April 27, 2016
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibitionHideyuki Igawa, Masashi Takahashi, Mikio Shirasaki, et al.Cytotherapy|October 25, 2024
Using qPCR and ddPCR to study biodistribution of cell therapy products: a multi-site evaluationEriko Fujita, Syunsuke Yamamoto, Takeshi Hanada, et al.Journal of Medicinal Chemistry|December 25, 2015
Structure-Based Design and Synthesis of 3-Amino-1,5-dihydro-4H-pyrazolopyridin-4-one Derivatives as Tyrosine Kinase 2 InhibitorsTakatoshi Yogo, Hiroyuki Nagamiya, Masaki Seto, et al.The Journal of Biological Chemistry|February 27, 2026
SLC52A1 Is a Neofunctionalized Primate Urate Transporter Enabling Intestinal Urate SecretionSyunsuke Yamamoto, Katsuhisa Inoue, Tomoya Yasujima, et al.Pageof 5