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Bioorganic & Medicinal Chemistry Letters|July 1, 2006
Hydrazides of clozapine: a new class of D1 dopamine receptor subtype selective antagonistsT K Sasikumar, D A Burnett, H Zhang, et al.Bioorganic & Medicinal Chemistry Letters|January 13, 2010
Remote functionalization of SCH 39166: discovery of potent and selective benzazepine dopamine D1 receptor antagonistsT K Sasikumar, Duane A Burnett, William J Greenlee, et al.Bioorganic & Medicinal Chemistry Letters|March 30, 2010
A-ring modifications on the triazafluorenone core structure and their mGluR1 antagonist propertiesT K Sasikumar, Li Qiang, Duane A Burnett, et al.Bioorganic & Medicinal Chemistry Letters|May 25, 2010
Tricyclic sulfones as orally active gamma-secretase inhibitors: synthesis and structure-activity relationship studiesT K Sasikumar, Li Qiang, Duane A Burnett, et al.Bioorganic & Medicinal Chemistry Letters|August 8, 2006
Novel aminobenzimidazoles as selective MCH-R1 antagonists for the treatment of metabolic diseasesT K Sasikumar, Li Qiang, Duane A Burnett, et al.Bioorganic & Medicinal Chemistry Letters|July 11, 2006
Tetrahydroisoquinolines as MCH-R1 antagonistsT K Sasikumar, L Qiang, W-L Wu, et al.Bioorganic & Medicinal Chemistry Letters|May 13, 2009
Tricyclic thienopyridine-pyrimidones/thienopyrimidine-pyrimidones as orally efficacious mGluR1 antagonists for neuropathic painT K Sasikumar, Li Qiang, Duane A Burnett, et al.Bioorganic & Medicinal Chemistry Letters|May 18, 2010
Tetracyclic sulfones as potent gamma-secretase inhibitors: synthesis and structure-activity relationship studiesT K Sasikumar, Duane A Burnett, Theodros Asberom, et al.Bioorganic & Medicinal Chemistry Letters|January 12, 2010
Discovery of new SCH 39166 analogs as potent and selective dopamine D1 receptor antagonistsLi Qiang, T K Sasikumar, Duane A Burnett, et al.Bioorganic & Medicinal Chemistry Letters|October 23, 2012
Synthesis and SAR development of novel mGluR1 antagonists for the treatment of chronic painStephanie Brumfield, Peter Korakas, Lisa S Silverman, et al.Pageof 1