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Organic & Biomolecular Chemistry|August 2, 2021
Fluorescence resonance energy transfer-based screening for protein kinase C ligands using 6-methoxynaphthalene-labeled 1,2-diacylglycerol-lactonesKohei Tsuji, Takahiro Ishii, Takuya Kobayakawa, et al.
Chembiochem : a European Journal of Chemical Biology|April 24, 2025
Hybrid Molecules of Small Molecular and Peptidic HIV Fusion InhibitorsKohei Tsuji, Takuya Kobayakawa, Peter Bolah, et al.
ACS Omega|October 20, 2025
SARS-CoV‑2 Papain-Like Protease Inhibitors Based on Naphthalen-1-ylethanamine and Halogenated Benzene MoietiesKouki Shinohara, Takuya Kobayakawa, Kohei Tsuji, et al.
European Journal of Medicinal Chemistry|October 23, 2024
Naphthalen-1-ylethanamine-containing small molecule inhibitors of the papain-like protease of SARS-CoV-2Kouki Shinohara, Takuya Kobayakawa, Kohei Tsuji, et al.
ACS Medicinal Chemistry Letters|January 20, 2018
Synthesis of a Chloroalkene Dipeptide Isostere-Containing Peptidomimetic and Its Biological ApplicationTakuya Kobayakawa, Yudai Matsuzaki, Kentaro Hozumi, et al.
Chembiochem : a European Journal of Chemical Biology|April 24, 2019
Dimeric C34 Derivatives Linked through Disulfide Bridges as New HIV-1 Fusion InhibitorsTakuya Kobayakawa, Kento Ebihara, Yuzuna Honda, et al.
Bioorganic & Medicinal Chemistry Letters|January 23, 2019
Soluble-type small-molecule CD4 mimics as HIV entry inhibitorsTakuya Kobayakawa, Kiju Konno, Nami Ohashi, et al.
The Journal of Organic Chemistry|March 18, 2021
Development of Methods for Convergent Synthesis of Chloroalkene Dipeptide Isosteres and Its ApplicationTakuya Kobayakawa, Chika Azuma, Yuki Watanabe, et al.
Organic & Biomolecular Chemistry|May 21, 2020
Synthesis of hydrophilic caged DAG-lactones for chemical biology applicationsTakuya Kobayakawa, Hikaru Takano, Takahiro Ishii, et al.
Journal of Medicinal Chemistry|December 15, 2025
Antibody-Drug Conjugates Using CD4 Mimics and a Neutralizing Antibody as HIV-1 Entry InhibitorsYutaro Miura, Kohei Tsuji, Takuya Kobayakawa, et al.
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