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Biochemistry|January 28, 2016
Characterization of the Enzymatic Activity of SETDB1 and Its 1:1 Complex with ATF7IPAravind Basavapathruni, Jodi Gureasko, Margaret Porter Scott, et al.The Journal of Biological Chemistry|August 13, 2010
SIRT1 activation by small molecules: kinetic and biophysical evidence for direct interaction of enzyme and activatorHan Dai, Lauren Kustigian, David Carney, et al.ACS Medicinal Chemistry Letters|July 21, 2022
Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical StudiesJoshua S Alford, John W Lampe, Dorothy Brach, et al.ACS Medicinal Chemistry Letters|October 21, 2021
Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical StudiesJohn W Lampe, Joshua S Alford, P Ann Boriak-Sjodin, et al.ACS Medicinal Chemistry Letters|March 18, 2016
Novel Oxindole Sulfonamides and Sulfamides: EPZ031686, the First Orally Bioavailable Small Molecule SMYD3 InhibitorLorna H Mitchell, P Ann Boriack-Sjodin, Sherri Smith, et al.Nature Communications|July 3, 2015
Crystallographic structure of a small molecule SIRT1 activator-enzyme complexHan Dai, April W Case, Thomas V Riera, et al.Science (New York, N.Y.)|March 9, 2013
Evidence for a common mechanism of SIRT1 regulation by allosteric activatorsBasil P Hubbard, Ana P Gomes, Han Dai, et al.Plos One|June 2, 2018
Small molecule inhibitors and CRISPR/Cas9 mutagenesis demonstrate that SMYD2 and SMYD3 activity are dispensable for autonomous cancer cell proliferationMichael J Thomenius, Jennifer Totman, Darren Harvey, et al.Pageof 2