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Organic Letters|April 27, 2002
Asymmetric synthesis of substituted prolines from delta-amino beta-ketoesters. Methyl (2S,5R)-(+)-5-phenylpyrrolidine-2-carboxylateFranklin A Davis, Tianan Fang, Rajesh GoswamiThe Journal of Organic Chemistry|October 25, 2001
Asymmetric Synthesis of 2H-Azirine 2-Carboxylate EstersFranklin A. Davis, Hu Liu, Chang-Hsing Liang, et al.Bioorganic & Medicinal Chemistry Letters|January 17, 2015
Pyridine and pyridinone-based factor XIa inhibitorsJames R Corte, Tianan Fang, Jon J Hangeland, et al.Steroids|April 10, 2004
Characterization of a new class of selective nonsteroidal progesterone receptor agonistsYu Dong, Jacques Y Roberge, Zhaoqing Wang, et al.Bioorganic & Medicinal Chemistry Letters|January 15, 2020
Orally bioavailable amine-linked macrocyclic inhibitors of factor XIaTianan Fang, James R Corte, Paul J Gilligan, et al.Journal of Medicinal Chemistry|January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide LinkerJames R Corte, Tianan Fang, Honey Osuna, et al.Bioorganic & Medicinal Chemistry|April 14, 2016
Orally bioavailable pyridine and pyrimidine-based Factor XIa inhibitors: Discovery of the methyl N-phenyl carbamate P2 prime groupJames R Corte, Tianan Fang, Donald J P Pinto, et al.Bioorganic & Medicinal Chemistry Letters|July 9, 2017
Macrocyclic inhibitors of Factor XIa: Discovery of alkyl-substituted macrocyclic amide linkers with improved potencyJames R Corte, Wu Yang, Tianan Fang, et al.Bioorganic & Medicinal Chemistry Letters|March 3, 2015
Structure-based design of inhibitors of coagulation factor XIa with novel P1 moietiesDonald J P Pinto, Joanne M Smallheer, James R Corte, et al.Bioorganic & Medicinal Chemistry Letters|April 22, 2008
Structure-activity relationships of anthranilamide-based factor Xa inhibitors containing piperidinone and pyridinone P4 moietiesJames R Corte, Tianan Fang, Donald J P Pinto, et al.Pageof 2