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ACS Medicinal Chemistry Letters
|
April 15, 2021
1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry
Silvio Aprile, Beatrice Riva, Irene Preet Bhela, et al.
Organic & Biomolecular Chemistry
|
April 16, 2011
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors
Margherita Guasconi, Xiaoyun Lu, Alberto Massarotti, et al.
Journal of Combinatorial Chemistry
|
July 5, 2008
Triazole-modified histone deacetylase inhibitors as a rapid route to drug discovery
Tracey Pirali, Francesca Pagliai, Ciro Mercurio, et al.
Molecular Diversity
|
May 29, 2009
Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition
Tracey Pirali, Valeria Faccio, Riccardo Mossetti, et al.
ACS Medicinal Chemistry Letters
|
December 20, 2023
Correction to "An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline"
Silvio Aprile, Giorgia Colombo, Marta Serafini, et al.
ACS Medicinal Chemistry Letters
|
August 18, 2022
An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline
Silvio Aprile, Giorgia Colombo, Marta Serafini, et al.
Chemmedchem
|
February 26, 2013
A concise synthesis of pyrazole analogues of combretastatin A1 as potent anti-tubulin agents
Roberta Zaninetti, Salvatore V Cortese, Silvio Aprile, et al.
Journal of Medicinal Chemistry
|
November 2, 2022
A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs
Irene Preet Bhela, Alice Ranza, Federica Carolina Balestrero, et al.
ACS Omega
|
February 17, 2025
Versatile One-Pot Synthesis of Hydrophobic Tags by Multicomponent Reactions
Federica Carolina Balestrero, Laura Gioiello, Georgia Goutsiou, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 6, 2018
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
Alessia Griglio, Enza Torre, Marta Serafini, et al.
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Search research articles
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Showing results (31-40 of 64) with videos related to
Sort By:
Page
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ACS Medicinal Chemistry Letters
|
April 15, 2021
1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry
Silvio Aprile, Beatrice Riva, Irene Preet Bhela, et al.
Organic & Biomolecular Chemistry
|
April 16, 2011
Groebke multicomponent reaction and subsequent nucleophilic aromatic substitution for a convenient synthesis of 3,8-diaminoimidazo[1,2-a]pyrazines as potential kinase inhibitors
Margherita Guasconi, Xiaoyun Lu, Alberto Massarotti, et al.
Journal of Combinatorial Chemistry
|
July 5, 2008
Triazole-modified histone deacetylase inhibitors as a rapid route to drug discovery
Tracey Pirali, Francesca Pagliai, Ciro Mercurio, et al.
Molecular Diversity
|
May 29, 2009
Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3+2] cycloaddition
Tracey Pirali, Valeria Faccio, Riccardo Mossetti, et al.
ACS Medicinal Chemistry Letters
|
December 20, 2023
Correction to "An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline"
Silvio Aprile, Giorgia Colombo, Marta Serafini, et al.
ACS Medicinal Chemistry Letters
|
August 18, 2022
An Unexpected Deuterium-Induced Metabolic Switch in Doxophylline
Silvio Aprile, Giorgia Colombo, Marta Serafini, et al.
Chemmedchem
|
February 26, 2013
A concise synthesis of pyrazole analogues of combretastatin A1 as potent anti-tubulin agents
Roberta Zaninetti, Salvatore V Cortese, Silvio Aprile, et al.
Journal of Medicinal Chemistry
|
November 2, 2022
A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs
Irene Preet Bhela, Alice Ranza, Federica Carolina Balestrero, et al.
ACS Omega
|
February 17, 2025
Versatile One-Pot Synthesis of Hydrophobic Tags by Multicomponent Reactions
Federica Carolina Balestrero, Laura Gioiello, Georgia Goutsiou, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 6, 2018
A multicomponent approach in the discovery of indoleamine 2,3-dioxygenase 1 inhibitors: Synthesis, biological investigation and docking studies
Alessia Griglio, Enza Torre, Marta Serafini, et al.
Page
of 7