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Journal of Medicinal Chemistry|December 3, 2025
Covalent Binding of the Boronic Acid-Based Inhibitor GSK4394835A to Phosphodiesterase 3B, a Drug Target for Cardiovascular DiseaseSamuel A Eaton, David W ChristiansonBiochemistry|December 21, 2006
Binding of uridine 5'-diphosphate in the "basic patch" of the zinc deacetylase LpxC and implications for substrate bindingHeather A Gennadios, David W ChristiansonPure and Applied Chemistry. Chimie Pure Et Appliquee|September 28, 2011
Trinuclear Metal Clusters in Catalysis by Terpenoid SynthasesJulie A Aaron, David W ChristiansonBiochemistry|February 29, 2024
Structure-Based Engineering of a Sesquiterpene Cyclase to Generate an Alcohol Product: Conversion of epi-Isozizaene Synthase into α-Bisabolol SynthaseSamuel A Eaton, David W ChristiansonJournal of the American Chemical Society|October 23, 2003
Design of amino acid sulfonamides as transition-state analogue inhibitors of arginaseEvis Cama, Hyunshun Shin, David W ChristiansonBiochemistry|November 21, 2019
Binding of N8-Acetylspermidine Analogues to Histone Deacetylase 10 Reveals Molecular Strategies for Blocking Polyamine DeacetylationCorey J Herbst-Gervasoni, David W ChristiansonBiochemistry|November 25, 2015
Structural Studies of Geosmin Synthase, a Bifunctional Sesquiterpene Synthase with αα Domain Architecture That Catalyzes a Unique Cyclization-Fragmentation Reaction SequenceGolda G Harris, Patrick M Lombardi, Travis A Pemberton, et al.Biochemistry|January 15, 2021
X-ray Crystallographic Snapshots of Substrate Binding in the Active Site of Histone Deacetylase 10Corey J Herbst-Gervasoni, David W ChristiansonJournal of the American Chemical Society|August 19, 2004
Design of amino acid aldehydes as transition-state analogue inhibitors of arginaseHyunshun Shin, Evis Cama, David W ChristiansonBioorganic & Medicinal Chemistry|June 25, 2013
Synthesis and evaluation of N⁸-acetylspermidine analogues as inhibitors of bacterial acetylpolyamine amidohydrolaseChristophe Decroos, Christine M Bowman, David W ChristiansonPageof 20