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Bioscience, Biotechnology, and Biochemistry
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November 28, 2022
Synthesis and structure-activity relationship study of aldose reductase inhibiting marine alkaloid lukianol A and its derivatives
Fumito Ishibashi, Shijiao Zha, Taiyo Kondo, et al.
Bioscience, Biotechnology, and Biochemistry
|
February 12, 2021
Concise synthesis and in vitro anticancer activity of benzo[g][1]benzopyrano[4,3-b]indol-6(13H)-ones (BBPIs), topoisomerase I inhibitors based on the marine alkaloid lamellarin
Fumito Ishibashi, Tsutomu Fukuda, Shijiao Zha, et al.
Bioorganic & Medicinal Chemistry
|
November 11, 2011
Synthesis, structure-activity relationships, and mechanism of action of anti-HIV-1 lamellarin α 20-sulfate analogues
Haruka Kamiyama, Yoshinao Kubo, Hironori Sato, et al.
Bioorganic & Medicinal Chemistry
|
December 17, 2018
Lamellarin-inspired potent topoisomerase I inhibitors with the unprecedented benzo[g][1]benzopyrano[4,3-b]indol-6(13H)-one scaffold
Tsutomu Fukuda, Yusuke Nanjo, Masahiro Fujimoto, et al.
Bioorganic & Medicinal Chemistry
|
November 15, 2017
Design, synthesis, and evaluation of A-ring-modified lamellarin N analogues as noncovalent inhibitors of the EGFR T790M/L858R mutant
Tsutomu Fukuda, Teppei Umeki, Keiji Tokushima, et al.
Bioorganic & Medicinal Chemistry
|
February 8, 2021
Synthesis and evaluation of azalamellarin N and its A-ring-modified analogues as non-covalent inhibitors of the EGFR T790M/L858R mutant
Tsutomu Fukuda, Mizuho Anzai, Akane Nakahara, et al.
Viruses
|
April 23, 2022
Unique Mode of Antiviral Action of a Marine Alkaloid against Ebola Virus and SARS-CoV-2
Mai Izumida, Osamu Kotani, Hideki Hayashi, et al.
Journal of Medicinal Chemistry
|
August 29, 2013
Synthesis, resolution, and biological evaluation of atropisomeric (aR)- and (aS)-16-methyllamellarins N: unique effects of the axial chirality on the selectivity of protein kinases inhibition
Kenyu Yoshida, Ryosuke Itoyama, Masashi Yamahira, et al.
Biological & Pharmaceutical Bulletin
|
January 3, 2024
Identification of Azalamellarin N as a Pyroptosis Inhibitor
Jun Takouda, Moeka Nakamura, Akane Murasaki, et al.
International Journal of Molecular Sciences
|
March 14, 2026
Development of a Conditional Replication System Using a Lassa Virus Glycoprotein Complex-Encoding Retroviral Vector for Isolating Resistant Variants to Inhibitors in BSL-2
Manya Bakatumana Hans, Anita Moendat Fanto, Tsutomu Fukuda, et al.
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Search research articles
Search
Showing results (11-20 of 22) with videos related to
Sort By:
Page
of 3
Bioscience, Biotechnology, and Biochemistry
|
November 28, 2022
Synthesis and structure-activity relationship study of aldose reductase inhibiting marine alkaloid lukianol A and its derivatives
Fumito Ishibashi, Shijiao Zha, Taiyo Kondo, et al.
Bioscience, Biotechnology, and Biochemistry
|
February 12, 2021
Concise synthesis and in vitro anticancer activity of benzo[g][1]benzopyrano[4,3-b]indol-6(13H)-ones (BBPIs), topoisomerase I inhibitors based on the marine alkaloid lamellarin
Fumito Ishibashi, Tsutomu Fukuda, Shijiao Zha, et al.
Bioorganic & Medicinal Chemistry
|
November 11, 2011
Synthesis, structure-activity relationships, and mechanism of action of anti-HIV-1 lamellarin α 20-sulfate analogues
Haruka Kamiyama, Yoshinao Kubo, Hironori Sato, et al.
Bioorganic & Medicinal Chemistry
|
December 17, 2018
Lamellarin-inspired potent topoisomerase I inhibitors with the unprecedented benzo[g][1]benzopyrano[4,3-b]indol-6(13H)-one scaffold
Tsutomu Fukuda, Yusuke Nanjo, Masahiro Fujimoto, et al.
Bioorganic & Medicinal Chemistry
|
November 15, 2017
Design, synthesis, and evaluation of A-ring-modified lamellarin N analogues as noncovalent inhibitors of the EGFR T790M/L858R mutant
Tsutomu Fukuda, Teppei Umeki, Keiji Tokushima, et al.
Bioorganic & Medicinal Chemistry
|
February 8, 2021
Synthesis and evaluation of azalamellarin N and its A-ring-modified analogues as non-covalent inhibitors of the EGFR T790M/L858R mutant
Tsutomu Fukuda, Mizuho Anzai, Akane Nakahara, et al.
Viruses
|
April 23, 2022
Unique Mode of Antiviral Action of a Marine Alkaloid against Ebola Virus and SARS-CoV-2
Mai Izumida, Osamu Kotani, Hideki Hayashi, et al.
Journal of Medicinal Chemistry
|
August 29, 2013
Synthesis, resolution, and biological evaluation of atropisomeric (aR)- and (aS)-16-methyllamellarins N: unique effects of the axial chirality on the selectivity of protein kinases inhibition
Kenyu Yoshida, Ryosuke Itoyama, Masashi Yamahira, et al.
Biological & Pharmaceutical Bulletin
|
January 3, 2024
Identification of Azalamellarin N as a Pyroptosis Inhibitor
Jun Takouda, Moeka Nakamura, Akane Murasaki, et al.
International Journal of Molecular Sciences
|
March 14, 2026
Development of a Conditional Replication System Using a Lassa Virus Glycoprotein Complex-Encoding Retroviral Vector for Isolating Resistant Variants to Inhibitors in BSL-2
Manya Bakatumana Hans, Anita Moendat Fanto, Tsutomu Fukuda, et al.
Page
of 3