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Methods in Molecular Biology (Clifton, N.J.)|March 31, 2025
Click Chemistry for Target Engagement StudiesSilvia Castelli, Sonia Troiani, Ulisse CucchiBiochemistry|August 7, 2013
Structural insight into maternal embryonic leucine zipper kinase (MELK) conformation and inhibition toward structure-based drug designGiulia Canevari, Stefania Re Depaolini, Ulisse Cucchi, et al.Molecular Cancer Therapeutics|September 18, 2023
Novel Thienoduocarmycin-Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical StudiesBarbara Valsasina, Paolo Orsini, Michele Caruso, et al.Science Translational Medicine|March 15, 2019
An antibody-drug conjugate directed to the ALK receptor demonstrates efficacy in preclinical models of neuroblastomaRenata Sano, Kateryna Krytska, Colleen E Larmour, et al.Anticancer Research|December 29, 2010
Phosphorylation of TCTP as a marker for polo-like kinase-1 activity in vivoUlisse Cucchi, Laura M Gianellini, Anna De Ponti, et al.Cancer Research|December 17, 2010
Targeting the mitotic checkpoint for cancer therapy with NMS-P715, an inhibitor of MPS1 kinaseRiccardo Colombo, Marina Caldarelli, Milena Mennecozzi, et al.Bioorganic & Medicinal Chemistry Letters|August 20, 2021
Identification of unprecedented ATP-competitive choline kinase inhibitorsFrancesca Quartieri, Marcella Nesi, Nilla R Avanzi, et al.Molecular Cancer Therapeutics|February 10, 2012
NMS-P937, an orally available, specific small-molecule polo-like kinase 1 inhibitor with antitumor activity in solid and hematologic malignanciesBarbara Valsasina, Italo Beria, Cristina Alli, et al.Nature Communications|June 10, 2017
A covalent PIN1 inhibitor selectively targets cancer cells by a dual mechanism of actionElena Campaner, Alessandra Rustighi, Alessandro Zannini, et al.Nature Chemical Biology|July 30, 2013
Covalent and allosteric inhibitors of the ATPase VCP/p97 induce cancer cell deathPaola Magnaghi, Roberto D'Alessio, Barbara Valsasina, et al.Pageof 1