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Chemmedchem|May 31, 2024
1,4-Pyrazolyl-Containing SAFit-Analogues are Selective FKBP51 Inhibitors With Improved Ligand Efficiency and Drug-Like ProfileVanessa Buffa, Christian Meyners, Wisely Oki Sugiarto, et al.
ACS Pharmacology & Translational Science|March 17, 2023
Analysis of the Selective Antagonist SAFit2 as a Chemical Probe for the FK506-Binding Protein 51Vanessa Buffa, Fabian H Knaup, Tim Heymann, et al.
Angewandte Chemie (International Ed. in English)|January 3, 2025
Conformational Plasticity and Binding Affinity Enhancement Controlled by Linker Derivatization in MacrocyclesVanessa Buffa, Carlo Walz, Christian Meyners, et al.
Communications Chemistry|December 4, 2025
Targeting bacterial kinases as a strategy to counteract antibiotic resistanceVanessa Buffa, Julien Kowalewski, Guoman Qi, et al.
Journal of Medicinal Chemistry|November 22, 2025
Linker Modification Enables Control of Key Functional Group Orientation in MacrocyclesChristian Brudy, Enrico Ruijsenaars, Christian Meyners, et al.
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