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Bioorganic & Medicinal Chemistry
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August 18, 2015
Heterocyclic chalcone activators of nuclear factor (erythroid-derived 2)-like 2 (Nrf2) with improved in vivo efficacy
Nicole Lounsbury, George Mateo, Brielle Jones, et al.
Journal of Chemical Information and Modeling
|
August 17, 2021
Discovery of Novel Small-Molecule Inhibitors of SARS-CoV-2 Main Protease as Potential Leads for COVID-19 Treatment
Anjela Manandhar, Vunnam Srinivasulu, Mohamad Hamad, et al.
Bioorganic & Medicinal Chemistry
|
January 30, 2008
Disruption of Kv1.1 N-type inactivation by novel small molecule inhibitors (disinactivators)
Qiang Lu, Joseph Peevey, Flora Jow, et al.
Leukemia & Lymphoma
|
October 3, 2018
Non-NAD-like PARP1 inhibitor enhanced synthetic lethal effect of NAD-like PARP inhibitors against BRCA1-deficient leukemia
Margaret Nieborowska-Skorska, Silvia Maifrede, Min Ye, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 26, 2009
Synthesis and structure-activity relationship of novel lactam-fused chroman derivatives having dual affinity at the 5-HT(1A) receptor and the serotonin transporter
Zhongqi Shen, P Siva Ramamoorthy, Nicole T Hatzenbuhler, et al.
Research Square
|
April 17, 2023
Haploinsufficiency of ZNF251 causes DNA-PKcs-dependent resistance to PARP inhibitors in BRCA1-mutated cancer cells
Huan Li, Srinivas Chatla, Xiaolei Liu, et al.
Bioorganic & Medicinal Chemistry
|
January 11, 2014
Synthesis and evaluation of Strychnos alkaloids as MDR reversal agents for cancer cell eradication
Surendrachary Munagala, Gopal Sirasani, Praveen Kokkonda, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 3, 2017
Design, synthesis and SAR of new-di-substituted pyridopyrimidines as ATP-competitive dual PI3Kα/mTOR inhibitors
Aisha A K Al-Ashmawy, Fatma A Ragab, Khaled M Elokely, et al.
Cancer Letters
|
February 1, 2025
ZNF251 haploinsufficiency confers PARP inhibitors resistance in BRCA1-mutated cancer cells through activation of homologous recombination
Huan Li, Srinivas Chatla, Xiaolei Liu, et al.
Blood
|
July 10, 2013
Personalized synthetic lethality induced by targeting RAD52 in leukemias identified by gene mutation and expression profile
Kimberly Cramer-Morales, Margaret Nieborowska-Skorska, Kara Scheibner, et al.
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of 4
Search research articles
Search
Showing results (21-30 of 35) with videos related to
Sort By:
Page
of 4
Bioorganic & Medicinal Chemistry
|
August 18, 2015
Heterocyclic chalcone activators of nuclear factor (erythroid-derived 2)-like 2 (Nrf2) with improved in vivo efficacy
Nicole Lounsbury, George Mateo, Brielle Jones, et al.
Journal of Chemical Information and Modeling
|
August 17, 2021
Discovery of Novel Small-Molecule Inhibitors of SARS-CoV-2 Main Protease as Potential Leads for COVID-19 Treatment
Anjela Manandhar, Vunnam Srinivasulu, Mohamad Hamad, et al.
Bioorganic & Medicinal Chemistry
|
January 30, 2008
Disruption of Kv1.1 N-type inactivation by novel small molecule inhibitors (disinactivators)
Qiang Lu, Joseph Peevey, Flora Jow, et al.
Leukemia & Lymphoma
|
October 3, 2018
Non-NAD-like PARP1 inhibitor enhanced synthetic lethal effect of NAD-like PARP inhibitors against BRCA1-deficient leukemia
Margaret Nieborowska-Skorska, Silvia Maifrede, Min Ye, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 26, 2009
Synthesis and structure-activity relationship of novel lactam-fused chroman derivatives having dual affinity at the 5-HT(1A) receptor and the serotonin transporter
Zhongqi Shen, P Siva Ramamoorthy, Nicole T Hatzenbuhler, et al.
Research Square
|
April 17, 2023
Haploinsufficiency of ZNF251 causes DNA-PKcs-dependent resistance to PARP inhibitors in BRCA1-mutated cancer cells
Huan Li, Srinivas Chatla, Xiaolei Liu, et al.
Bioorganic & Medicinal Chemistry
|
January 11, 2014
Synthesis and evaluation of Strychnos alkaloids as MDR reversal agents for cancer cell eradication
Surendrachary Munagala, Gopal Sirasani, Praveen Kokkonda, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 3, 2017
Design, synthesis and SAR of new-di-substituted pyridopyrimidines as ATP-competitive dual PI3Kα/mTOR inhibitors
Aisha A K Al-Ashmawy, Fatma A Ragab, Khaled M Elokely, et al.
Cancer Letters
|
February 1, 2025
ZNF251 haploinsufficiency confers PARP inhibitors resistance in BRCA1-mutated cancer cells through activation of homologous recombination
Huan Li, Srinivas Chatla, Xiaolei Liu, et al.
Blood
|
July 10, 2013
Personalized synthetic lethality induced by targeting RAD52 in leukemias identified by gene mutation and expression profile
Kimberly Cramer-Morales, Margaret Nieborowska-Skorska, Kara Scheibner, et al.
Page
of 4