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Nature Biotechnology
|
January 7, 2022
Conformation-locking antibodies for the discovery and characterization of KRAS inhibitors
Christopher W Davies, Angela J Oh, Rana Mroue, et al.
ACS Medicinal Chemistry Letters
|
December 30, 2015
Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety
Chudi O Ndubaku, James J Crawford, Joy Drobnick, et al.
Cancer Cell
|
December 8, 2009
Somatic mutations in p85alpha promote tumorigenesis through class IA PI3K activation
Bijay S Jaiswal, Vasantharajan Janakiraman, Noelyn M Kljavin, et al.
Journal of Medicinal Chemistry
|
January 11, 2014
Fragment-based identification of amides derived from trans-2-(pyridin-3-yl)cyclopropanecarboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
Anthony M Giannetti, Xiaozhang Zheng, Nicholas J Skelton, et al.
ACS Medicinal Chemistry Letters
|
January 21, 2022
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1)
Bryan K Chan, Eileen Seward, Michael Lainchbury, et al.
ACS Medicinal Chemistry Letters
|
September 18, 2024
Discovery of GNE-6893, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of HPK1
John C Tellis, BinQing Wei, Michael Siu, et al.
Journal of Medicinal Chemistry
|
July 18, 2013
Structure-based discovery of novel amide-containing nicotinamide phosphoribosyltransferase (nampt) inhibitors
Xiaozhang Zheng, Paul Bauer, Timm Baumeister, et al.
Journal of Medicinal Chemistry
|
May 12, 2016
Chemically Diverse Group I p21-Activated Kinase (PAK) Inhibitors Impart Acute Cardiovascular Toxicity with a Narrow Therapeutic Window
Joachim Rudolph, Lesley J Murray, Chudi O Ndubaku, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 4, 2015
Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility
Mark Zak, Bianca M Liederer, Deepak Sampath, et al.
Nature
|
August 17, 2012
Recurrent R-spondin fusions in colon cancer
Somasekar Seshagiri, Eric W Stawiski, Steffen Durinck, et al.
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Search research articles
Search
Showing results (71-80 of 91) with videos related to
Sort By:
Page
of 10
Nature Biotechnology
|
January 7, 2022
Conformation-locking antibodies for the discovery and characterization of KRAS inhibitors
Christopher W Davies, Angela J Oh, Rana Mroue, et al.
ACS Medicinal Chemistry Letters
|
December 30, 2015
Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety
Chudi O Ndubaku, James J Crawford, Joy Drobnick, et al.
Cancer Cell
|
December 8, 2009
Somatic mutations in p85alpha promote tumorigenesis through class IA PI3K activation
Bijay S Jaiswal, Vasantharajan Janakiraman, Noelyn M Kljavin, et al.
Journal of Medicinal Chemistry
|
January 11, 2014
Fragment-based identification of amides derived from trans-2-(pyridin-3-yl)cyclopropanecarboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
Anthony M Giannetti, Xiaozhang Zheng, Nicholas J Skelton, et al.
ACS Medicinal Chemistry Letters
|
January 21, 2022
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1)
Bryan K Chan, Eileen Seward, Michael Lainchbury, et al.
ACS Medicinal Chemistry Letters
|
September 18, 2024
Discovery of GNE-6893, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of HPK1
John C Tellis, BinQing Wei, Michael Siu, et al.
Journal of Medicinal Chemistry
|
July 18, 2013
Structure-based discovery of novel amide-containing nicotinamide phosphoribosyltransferase (nampt) inhibitors
Xiaozhang Zheng, Paul Bauer, Timm Baumeister, et al.
Journal of Medicinal Chemistry
|
May 12, 2016
Chemically Diverse Group I p21-Activated Kinase (PAK) Inhibitors Impart Acute Cardiovascular Toxicity with a Narrow Therapeutic Window
Joachim Rudolph, Lesley J Murray, Chudi O Ndubaku, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 4, 2015
Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility
Mark Zak, Bianca M Liederer, Deepak Sampath, et al.
Nature
|
August 17, 2012
Recurrent R-spondin fusions in colon cancer
Somasekar Seshagiri, Eric W Stawiski, Steffen Durinck, et al.
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of 10