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Bioorganic & Medicinal Chemistry Letters|June 11, 2016
Alkyl substituted aminal derivatives of HCV NS5A inhibitor MK-8742Wensheng Yu, Craig A Coburn, Anilkumar G Nair, et al.Bioorganic & Medicinal Chemistry Letters|February 7, 2016
Discovery of silyl proline containing HCV NS5A inhibitors with pan-genotype activity: SAR developmentAnilkumar G Nair, Qingbei Zeng, Oleg Selyutin, et al.Bioorganic & Medicinal Chemistry Letters|November 26, 2010
Novel TNF-α converting enzyme (TACE) inhibitors as potential treatment for inflammatory diseasesVinay M Girijavallabhan, Lei Chen, Chaoyang Dai, et al.Journal of Medicinal Chemistry|February 18, 2014
The discovery of N-((2H-tetrazol-5-yl)methyl)-4-((R)-1-((5r,8R)-8-(tert-butyl)-3-(3,5-dichlorophenyl)-2-oxo-1,4-diazaspiro[4.5]dec-3-en-1-yl)-4,4-dimethylpentyl)benzamide (SCH 900822): a potent and selective glucagon receptor antagonistDuane DeMong, Xing Dai, Joyce Hwa, et al.Bioorganic & Medicinal Chemistry Letters|December 22, 2009
The discovery of novel tartrate-based TNF-alpha converting enzyme (TACE) inhibitorsKristin E Rosner, Zhuyan Guo, Peter Orth, et al.Bioorganic & Medicinal Chemistry Letters|July 20, 2010
Structure and activity relationships of tartrate-based TACE inhibitorsDansu Li, Janeta Popovici-Muller, David B Belanger, et al.Bioorganic & Medicinal Chemistry Letters|August 3, 2020
Potent, non-covalent reversible BTK inhibitors with 8-amino-imidazo[1,5-a]pyrazine core featuring 3-position bicyclic ring substitutesJian Liu, Deodial Guiadeen, Arto Krikorian, et al.ACS Medicinal Chemistry Letters|March 19, 2021
Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 InhibitorsDerun Li, Yongqi Deng, Abdelghani Achab, et al.Pageof 13