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Journal of Medicinal Chemistry
|
February 1, 2008
Malaria-infected mice are cured by oral administration of new artemisinin derivatives
Gary H Posner, Wonsuk Chang, Lindsey Hess, et al.
Antimicrobial Agents and Chemotherapy
|
March 31, 2010
Preclinical evaluation of the antifolate QN254, 5-chloro- N'6'-(2,5-dimethoxy-benzyl)-quinazoline-2,4,6-triamine, as an antimalarial drug candidate
Alexis Nzila, Matthias Rottmann, Penchit Chitnumsub, et al.
ACS Infectious Diseases
|
September 11, 2023
Antimalarial Dibenzannulated Medium-Ring Keto Lactams
Rongguo Ren, Xiaofang Wang, Derek A Leas, et al.
Chemmedchem
|
September 21, 2022
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2
Benoît Laleu, Kelly Rubiano, Tomas Yeo, et al.
ACS Omega
|
April 22, 2022
Metabolic, Pharmacokinetic, and Activity Profile of the Liver Stage Antimalarial (RC-12)
Yuxiang Dong, Yogesh Sonawane, Steven P Maher, et al.
Journal of Medicinal Chemistry
|
April 19, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ <sup>null</sup> Mouse Model of Malaria
Aloysius T Nchinda, Claire Le Manach, Tanya Paquet, et al.
Journal of Medicinal Chemistry
|
August 26, 2021
Discovery and Structure-Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials
Benoît Laleu, Yuichiro Akao, Atsuko Ochida, et al.
Journal of Medicinal Chemistry
|
November 30, 2012
Structure-activity relationship studies of orally active antimalarial 3,5-substituted 2-aminopyridines
Diego González Cabrera, Frederic Douelle, Yassir Younis, et al.
Journal of Medicinal Chemistry
|
March 19, 2015
Inhibitors of plasmodial serine hydroxymethyltransferase (SHMT): cocrystal structures of pyrazolopyrans with potent blood- and liver-stage activities
Matthias C Witschel, Matthias Rottmann, Anatol Schwab, et al.
Journal of Medicinal Chemistry
|
February 23, 2021
Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in <i>Plasmodium falciparum</i>
Aloysus Lawong, Suraksha Gahalawat, John Okombo, et al.
Page
of 32
Search research articles
Search
Showing results (231-240 of 318) with videos related to
Sort By:
Page
of 32
Journal of Medicinal Chemistry
|
February 1, 2008
Malaria-infected mice are cured by oral administration of new artemisinin derivatives
Gary H Posner, Wonsuk Chang, Lindsey Hess, et al.
Antimicrobial Agents and Chemotherapy
|
March 31, 2010
Preclinical evaluation of the antifolate QN254, 5-chloro- N'6'-(2,5-dimethoxy-benzyl)-quinazoline-2,4,6-triamine, as an antimalarial drug candidate
Alexis Nzila, Matthias Rottmann, Penchit Chitnumsub, et al.
ACS Infectious Diseases
|
September 11, 2023
Antimalarial Dibenzannulated Medium-Ring Keto Lactams
Rongguo Ren, Xiaofang Wang, Derek A Leas, et al.
Chemmedchem
|
September 21, 2022
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2
Benoît Laleu, Kelly Rubiano, Tomas Yeo, et al.
ACS Omega
|
April 22, 2022
Metabolic, Pharmacokinetic, and Activity Profile of the Liver Stage Antimalarial (RC-12)
Yuxiang Dong, Yogesh Sonawane, Steven P Maher, et al.
Journal of Medicinal Chemistry
|
April 19, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ <sup>null</sup> Mouse Model of Malaria
Aloysius T Nchinda, Claire Le Manach, Tanya Paquet, et al.
Journal of Medicinal Chemistry
|
August 26, 2021
Discovery and Structure-Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials
Benoît Laleu, Yuichiro Akao, Atsuko Ochida, et al.
Journal of Medicinal Chemistry
|
November 30, 2012
Structure-activity relationship studies of orally active antimalarial 3,5-substituted 2-aminopyridines
Diego González Cabrera, Frederic Douelle, Yassir Younis, et al.
Journal of Medicinal Chemistry
|
March 19, 2015
Inhibitors of plasmodial serine hydroxymethyltransferase (SHMT): cocrystal structures of pyrazolopyrans with potent blood- and liver-stage activities
Matthias C Witschel, Matthias Rottmann, Anatol Schwab, et al.
Journal of Medicinal Chemistry
|
February 23, 2021
Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in <i>Plasmodium falciparum</i>
Aloysus Lawong, Suraksha Gahalawat, John Okombo, et al.
Page
of 32