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Expert Opinion on Drug Discovery
|
August 30, 2025
Advances in click chemistry for drug discovery and development
Jiaojiao Dai, Xiaojia Xue, Xiangyi Jiang, et al.
Expert Opinion on Drug Discovery
|
May 17, 2019
Recent applications of click chemistry in drug discovery
Xiangyi Jiang, Xia Hao, Lanlan Jing, et al.
Drug Discovery Today
|
July 1, 2024
Recent advances in the molecular design and applications of viral RNA-targeting antiviral modalities
Jiaojiao Dai, Xiangyi Jiang, Edeildo Ferreira da Silva-Júnior, et al.
Expert Opinion on Drug Discovery
|
December 8, 2022
The discovery and design of novel HIV-1 capsid modulators and future perspectives
Dang Ding, Shujing Xu, Xujie Zhang, et al.
Expert Opinion on Drug Discovery
|
November 21, 2023
Advances in drug structure-activity-relationships for the development of selenium-based compounds against HIV
Dazhou Shi, Shujing Xu, Dang Ding, et al.
Journal of Medicinal Chemistry
|
January 8, 2026
First-in-Class Quinoline-Dione-Derived PROTACs: Potent Degraders of Cdc25 Phosphatases for Antitumor Therapy
Guanyu Dong, Mengfei Chen, Xiangyi Jiang, et al.
European Journal of Medicinal Chemistry
|
November 13, 2024
Discovery of novel fused-heterocycle-bearing diarypyrimidine derivatives as HIV-1 potent NNRTIs targeting tolerant region I for enhanced antiviral activity and resistance profile
Jiaojiao Dai, Xiangyi Jiang, Heng Gao, et al.
Journal of Medicinal Chemistry
|
October 20, 2025
Structure- and Privileged Fragment-Based Iterative Optimization: Discovery of 2,4-Disubstituted-6-aminopyrimidines as Novel HIV-1 NNRTIs with Potent Activity against Drug-Resistant Strains and Favorable Safety Profiles
Xiangkai Ji, Xiangyi Jiang, Heng Gao, et al.
Journal of Medicinal Chemistry
|
August 25, 2021
Discovery of Novel Dihydrothiopyrano[4,3-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 NNRTIs with Significantly Reduced hERG Inhibitory Activity and Improved Resistance Profiles
Zhao Wang, Waleed A Zalloum, Wenbo Wang, et al.
European Journal of Medicinal Chemistry
|
September 25, 2020
Targeting dual tolerant regions of binding pocket: Discovery of novel morpholine-substituted diarylpyrimidines as potent HIV-1 NNRTIs with significantly improved water solubility
Zhao Wang, Dongwei Kang, Da Feng, et al.
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Search research articles
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Showing results (1-10 of 45) with videos related to
Sort By:
Page
of 5
Expert Opinion on Drug Discovery
|
August 30, 2025
Advances in click chemistry for drug discovery and development
Jiaojiao Dai, Xiaojia Xue, Xiangyi Jiang, et al.
Expert Opinion on Drug Discovery
|
May 17, 2019
Recent applications of click chemistry in drug discovery
Xiangyi Jiang, Xia Hao, Lanlan Jing, et al.
Drug Discovery Today
|
July 1, 2024
Recent advances in the molecular design and applications of viral RNA-targeting antiviral modalities
Jiaojiao Dai, Xiangyi Jiang, Edeildo Ferreira da Silva-Júnior, et al.
Expert Opinion on Drug Discovery
|
December 8, 2022
The discovery and design of novel HIV-1 capsid modulators and future perspectives
Dang Ding, Shujing Xu, Xujie Zhang, et al.
Expert Opinion on Drug Discovery
|
November 21, 2023
Advances in drug structure-activity-relationships for the development of selenium-based compounds against HIV
Dazhou Shi, Shujing Xu, Dang Ding, et al.
Journal of Medicinal Chemistry
|
January 8, 2026
First-in-Class Quinoline-Dione-Derived PROTACs: Potent Degraders of Cdc25 Phosphatases for Antitumor Therapy
Guanyu Dong, Mengfei Chen, Xiangyi Jiang, et al.
European Journal of Medicinal Chemistry
|
November 13, 2024
Discovery of novel fused-heterocycle-bearing diarypyrimidine derivatives as HIV-1 potent NNRTIs targeting tolerant region I for enhanced antiviral activity and resistance profile
Jiaojiao Dai, Xiangyi Jiang, Heng Gao, et al.
Journal of Medicinal Chemistry
|
October 20, 2025
Structure- and Privileged Fragment-Based Iterative Optimization: Discovery of 2,4-Disubstituted-6-aminopyrimidines as Novel HIV-1 NNRTIs with Potent Activity against Drug-Resistant Strains and Favorable Safety Profiles
Xiangkai Ji, Xiangyi Jiang, Heng Gao, et al.
Journal of Medicinal Chemistry
|
August 25, 2021
Discovery of Novel Dihydrothiopyrano[4,3-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 NNRTIs with Significantly Reduced hERG Inhibitory Activity and Improved Resistance Profiles
Zhao Wang, Waleed A Zalloum, Wenbo Wang, et al.
European Journal of Medicinal Chemistry
|
September 25, 2020
Targeting dual tolerant regions of binding pocket: Discovery of novel morpholine-substituted diarylpyrimidines as potent HIV-1 NNRTIs with significantly improved water solubility
Zhao Wang, Dongwei Kang, Da Feng, et al.
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of 5