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European Journal of Medicinal Chemistry|March 28, 2024
Discovery of novel and selective farnesoid X receptor antagonists through structure-based virtual screening, preliminary structure-activity relationship study, and biological evaluationXiaodong Dou, Tongyu Huo, Yameng Liu, et al.Journal of the American Chemical Society|July 15, 2022
Catalytic Electrophilic Halogenation of Arenes with Electron-Withdrawing SubstituentsWeijin Wang, Xiaoxue Yang, Rongheng Dai, et al.European Journal of Medicinal Chemistry|February 10, 2023
The structure-based optimization of 3-substituted indolin-2-one derivatives as potent and isoform-selective c-Jun N-terminal kinase 3 (JNK3) inhibitors and biological evaluationZhongtang Li, Guiwang Zhu, Xiaoang Liu, et al.European Journal of Medicinal Chemistry|December 18, 2018
Unravel a neuroactive sHA sulfation pattern with neurogenesis activity by a library of defined oligosaccharidesWang Yao, Man Chen, Xiaodong Dou, et al.Bioorganic & Medicinal Chemistry Letters|November 9, 2023
Discovery of 3-oxo-1,2,3,4-tetrahydropyrido[1,2-a]pyrazin derivatives as SARS-CoV-2 main protease inhibitors through virtual screening and biological evaluationXiaodong Dou, Qi Sun, Yameng Liu, et al.European Journal of Medicinal Chemistry|March 1, 2022
Discovery of novel ataxia telangiectasia mutated (ATM) kinase modulators: Computational simulation, biological evaluation and cancer combinational chemotherapy studyXiaodong Dou, Xiaojiao Sun, Huixia Huang, et al.Acta Pharmaceutica Sinica. B|June 29, 2026
Discovery of sulfonyl benzoic acid derivatives with joint TGR5-agonist and FXR-antagonist activity for myocardial ischemia/reperfusion injury protectionXinyi Zhao, Tianqi Chang, Xiang Wu, et al.European Journal of Medicinal Chemistry|June 10, 2022
Discovery of 2-(furan-2-ylmethylene)hydrazine-1-carbothioamide derivatives as novel inhibitors of SARS-CoV-2 main proteaseXiaodong Dou, Qi Sun, Guofeng Xu, et al.Pageof 2