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International Journal of Molecular Sciences|January 25, 2025
Optimization of SARS-CoV-2 Mpro Inhibitors by a Structure-Based Multilevel Virtual Screening MethodLanlan Jing, Fabao Zhao, Lin Zheng, et al.Bioorganic & Medicinal Chemistry|August 10, 2016
Arylazolyl(azinyl)thioacetanilides. Part 20: Discovery of novel purinylthioacetanilides derivatives as potent HIV-1 NNRTIs via a structure-based bioisosterism approachXueyi Lu, Xiao Li, Jiapei Yang, et al.Journal of Medicinal Chemistry|June 20, 2018
Identification of Potent Ebola Virus Entry Inhibitors with Suitable Properties for in Vivo StudiesHu Liu, Ye Tian, Kyungae Lee, et al.European Journal of Medicinal Chemistry|October 18, 2016
Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangementXiao Li, Ping Gao, Boshi Huang, et al.Journal of Molecular Biology|February 26, 2022
Novel RNase H Inhibitors Blocking RNA-directed Strand Displacement DNA Synthesis by HIV-1 Reverse TranscriptaseSamara Martín-Alonso, Dongwei Kang, Javier Martínez Del Río, et al.Journal of Medicinal Chemistry|September 17, 2025
Exploring the HIV-1 Reverse Transcriptase p51/p66 Interface: Structure-Based Design and Optimization of Novel 2,4,6-Trisubstituted Pyrimidines as Potent NNRTIs with Improved Resistance ProfilesXiangkai Ji, Xiangyi Jiang, Zhen Gao, et al.Bioorganic & Medicinal Chemistry|June 30, 2017
Discovery of novel DAPY-IAS hybrid derivatives as potential HIV-1 inhibitors using molecular hybridization based on crystallographic overlaysBoshi Huang, Xueshun Wang, Xinhao Liu, et al.European Journal of Medicinal Chemistry|March 6, 2025
Structure-based design of novel 2,4,5-trisubstituted pyrimidine derivatives as potent HIV-1 NNRTIs by exploiting the tolerant regions in NNTRIs binding pocketZhenzhen Zhou, Minghui Xie, Zongji Zhuo, et al.Journal of Medicinal Chemistry|July 18, 2025
Probing the Dominant Motifs within the Hydrophobic Channel Yields Oxadiazole-Containing Diarylpyrimidine Derivatives as Potent HIV-1 Non-Nucleoside Reverse Transcriptase InhibitorsTao Zhang, Yue Yang, Xin Li, et al.Bioorganic Chemistry|August 24, 2021
Discovery of potent and selective Cdc25 phosphatase inhibitors via rapid assembly and in situ screening of Quinonoid-focused librariesYucen Tao, Xia Hao, Lanlan Jing, et al.Pageof 40