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Journal of Medicinal Chemistry
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August 10, 2018
Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101)
Yosup Rew, Xiaohui Du, John Eksterowicz, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 3, 2009
Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11 beta-HSD1 inhibitors
Dustin L McMinn, Yosup Rew, Athena Sudom, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 26, 2010
The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors
Xuelei Yan, Zhulun Wang, Athena Sudom, et al.
Journal of Medicinal Chemistry
|
June 17, 2008
Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model
Lisa D Julian, Zhulun Wang, Tracy Bostick, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 25, 2010
Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
Daqing Sun, Zhulun Wang, Seb Caille, et al.
Journal of Medicinal Chemistry
|
March 28, 2020
Discovery of Potent and Selective Non-Nucleotide Small Molecule Inhibitors of CD73
Joel W Beatty, Erick A Lindsey, Rhiannon Thomas-Tran, et al.
Journal of Medicinal Chemistry
|
April 29, 2026
Discovery of Casdatifan, Part I: Design and Characterization of Tetrahydroquinoline Inhibitors of Hypoxia-Inducible Factor-2α
Guillaume Mata, Artur K Mailyan, Samuel L Drew, et al.
ACS Medicinal Chemistry Letters
|
August 23, 2014
Discovery of Potent and Simplified Piperidinone-Based Inhibitors of the MDM2-p53 Interaction
Ming Yu, Yingcai Wang, Jiang Zhu, et al.
Journal of Medicinal Chemistry
|
November 19, 2019
Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere
Gwenaella Rescourio, Ana Z Gonzalez, Salman Jabri, et al.
ACS Medicinal Chemistry Letters
|
November 20, 2020
Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors
Dillon H Miles, Xuelei Yan, Rhiannon Thomas-Tran, et al.
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of 4
Search research articles
Search
Showing results (21-30 of 39) with videos related to
Sort By:
Page
of 4
Journal of Medicinal Chemistry
|
August 10, 2018
Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101)
Yosup Rew, Xiaohui Du, John Eksterowicz, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 3, 2009
Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11 beta-HSD1 inhibitors
Dustin L McMinn, Yosup Rew, Athena Sudom, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 26, 2010
The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors
Xuelei Yan, Zhulun Wang, Athena Sudom, et al.
Journal of Medicinal Chemistry
|
June 17, 2008
Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model
Lisa D Julian, Zhulun Wang, Tracy Bostick, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 25, 2010
Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
Daqing Sun, Zhulun Wang, Seb Caille, et al.
Journal of Medicinal Chemistry
|
March 28, 2020
Discovery of Potent and Selective Non-Nucleotide Small Molecule Inhibitors of CD73
Joel W Beatty, Erick A Lindsey, Rhiannon Thomas-Tran, et al.
Journal of Medicinal Chemistry
|
April 29, 2026
Discovery of Casdatifan, Part I: Design and Characterization of Tetrahydroquinoline Inhibitors of Hypoxia-Inducible Factor-2α
Guillaume Mata, Artur K Mailyan, Samuel L Drew, et al.
ACS Medicinal Chemistry Letters
|
August 23, 2014
Discovery of Potent and Simplified Piperidinone-Based Inhibitors of the MDM2-p53 Interaction
Ming Yu, Yingcai Wang, Jiang Zhu, et al.
Journal of Medicinal Chemistry
|
November 19, 2019
Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere
Gwenaella Rescourio, Ana Z Gonzalez, Salman Jabri, et al.
ACS Medicinal Chemistry Letters
|
November 20, 2020
Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors
Dillon H Miles, Xuelei Yan, Rhiannon Thomas-Tran, et al.
Page
of 4