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ACS Medicinal Chemistry Letters|May 22, 2020
A Class of Potent Inhibitors of the HIV-1 Nucleocapsid Protein Based on Aminopyrrolic ScaffoldsStefano Ciaco, Nicolas Humbert, Eléonore Real, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
New Dual CK2/HDAC1 Inhibitors with Nanomolar Inhibitory Activity against Both EnzymesLoganathan Rangasamy, Irene Ortín, José María Zapico, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Developing Cyclic Opioid Analogues: Fluorescently Labeled Bioconjugates of BiphalinAzzurra Stefanucci, Marilisa Pia Dimmito, Gabriela Molnar, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole InhibitorsJessica Caciolla, Angelo Spinello, Silvia Martini, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Pharmacophore-Based Design of New Chemical Scaffolds as Translational Readthrough-Inducing Drugs (TRIDs)Marco Tutone, Ivana Pibiri, Riccardo Perriera, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid ProteinSavina Malancona, Mattia Mori, Paola Fezzardi, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 PolymeraseRolando Cannalire, Kitti Wing Ki Chan, Maria Sole Burali, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Drug Synergism: Studies of Combination of RK-52 and Curcumin against Rhodesain of Trypanosoma brucei rhodesienseRoberta Ettari, Santo Previti, Carla Di Chio, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
From PARP1 to TNKS2 Inhibition: A Structure-Based ApproachStefano Tomassi, Julian Pfahler, Nicola Mautone, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Synthesis of Novel G Factor or Chloroquine-Artemisinin Hybrids and Conjugates with Potent Antiplasmodial ActivityDionissia A Pepe, Dimitra Toumpa, Christiane André-Barrès, et al.
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