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ACS Medicinal Chemistry Letters|March 18, 2016
Epigenetic Medicinal ChemistryRobert A Copeland
ACS Medicinal Chemistry Letters|March 18, 2016
Characterizing the Covalent Targets of a Small Molecule Inhibitor of the Lysine Acetyltransferase P300Jonathan H Shrimp, Alexander W Sorum, Julie M Garlick, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Design and Synthesis of Nonpeptide Inhibitors of Hepatocyte Growth Factor ActivationPhanindra K M Venukadasula, Benjamin Y Owusu, Namita Bansal, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 AgonistsGuido Galley, Angélica Beurier, Guillaume Décoret, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Discovery of 8-Amino-imidazo[1,5-a]pyrazines as Reversible BTK Inhibitors for the Treatment of Rheumatoid ArthritisJian Liu, Deodial Guiadeen, Arto Krikorian, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Discovery of a Novel 2,6-Disubstituted Glucosamine Series of Potent and Selective Hexokinase 2 InhibitorsHong Lin, Jin Zeng, Ren Xie, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Development of a Potent, Specific CDK8 Kinase Inhibitor Which Phenocopies CDK8/19 Knockout CellsMichael F T Koehler, Philippe Bergeron, Elizabeth M Blackwood, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Structure-Activity Relationship Studies and Molecular Modeling of Naphthalene-Based Sphingosine Kinase 2 InhibitorsMolly D Congdon, Yugesh Kharel, Anne M Brown, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Design, Syntheses, and Anti-TB Activity of 1,3-Benzothiazinone Azide and Click Chemistry Products Inspired by BTZ043Rohit Tiwari, Patricia A Miller, Laurent R Chiarelli, et al.
ACS Medicinal Chemistry Letters|March 18, 2016
Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical TrialsT G Murali Dhar, Hai-Yun Xiao, Jenny Xie, et al.
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