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ACS Medicinal Chemistry Letters|March 21, 2019
Use of a Conformational-Switching Mechanism to Modulate Exposed Polarity: Discovery of CCR2 Antagonist BMS-741672Michael G Yang, Zili Xiao, Robert J Cherney, et al.ACS Medicinal Chemistry Letters|March 21, 2019
Enhancing Drug Residence Time by Shielding of Intra-Protein Hydrogen Bonds: A Case Study on CCR2 AntagonistsAniket Magarkar, Gisela Schnapp, Anna-Katharina Apel, et al.ACS Medicinal Chemistry Letters|March 21, 2019
Discovery of Soft-Drug Topical Tool Modulators of Sphingosine-1-phosphate Receptor 1 (S1PR1)Mark Bell, David Foley, Claire Naylor, et al.ACS Medicinal Chemistry Letters|March 21, 2019
Second Generation Inhibitors of HIV-1 MaturationAlicia Regueiro-Ren, Ira B Dicker, Umesh Hanumegowda, et al.ACS Medicinal Chemistry Letters|April 25, 2017
RITA Mimics: Synthesis and Mechanistic Evaluation of Asymmetric Linked TrithiazolesAdrian L Pietkiewicz, Yuqi Zhang, Marwa N Rahimi, et al.ACS Medicinal Chemistry Letters|April 25, 2017
18F-Labeled Pyrido[3,4-d]pyrimidine as an Effective Probe for Imaging of L858R Mutant Epidermal Growth Factor ReceptorHiroyuki Kimura, Haruka Okuda, Masumi Ishiguro, et al.ACS Medicinal Chemistry Letters|April 25, 2017
Discovery of the First Environment-Sensitive Fluorescent Probe for GPR120 (FFA4) ImagingJiaxiang Liu, Chengsen Tian, Tianyu Jiang, et al.ACS Medicinal Chemistry Letters|April 25, 2017
Opioid Receptor Activity and Analgesic Potency of DPDPE Peptide Analogues Containing a Xylene BridgeAzzurra Stefanucci, Ettore Novellino, Sako Mirzaie, et al.ACS Medicinal Chemistry Letters|April 25, 2017
Norbenzomorphan Scaffold: Chemical Tool for Modulating Sigma Receptor-Subtype SelectivityJames J Sahn, Timothy R Hodges, Jessica Z Chan, et al.ACS Medicinal Chemistry Letters|March 21, 2019
Discovery of a JAK1/3 Inhibitor and Use of a Prodrug To Demonstrate Efficacy in a Model of Rheumatoid ArthritisSteven H Spergel, Michael E Mertzman, James Kempson, et al.Pageof 438