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ACS Medicinal Chemistry Letters|May 15, 2024
Identification of Dual Inhibitors Targeting Main Protease (Mpro) and Cathepsin L as Potential Anti-SARS-CoV-2 AgentsSanto Previti, Roberta Ettari, Elsa Calcaterra, et al.ACS Medicinal Chemistry Letters|May 15, 2024
Structural Investigations of Phthalazinone Derivatives as Allosteric Inhibitors of Human DNA Methyltransferase 3AIvan Hernandez, Ethan Ward, Thomas R R Pettus, et al.ACS Medicinal Chemistry Letters|May 15, 2024
Discovery of Novel Bicyclic Pyrazoles as Potent PIP5K1C InhibitorsKoji Ochiai, Shigeki Seto, Masanobu Yajima, et al.ACS Medicinal Chemistry Letters|May 15, 2024
Simple Fluorescence Labeling Method Enables Detection of Intracellular Distribution and Expression Level of Retinoid X ReceptorsYukina Tanaka, Michiko Fujihara, Yuta Takamura, et al.ACS Medicinal Chemistry Letters|April 17, 2024
Chemical Space Profiling of SARS-CoV-2 PLpro Using DNA-Encoded Focused LibrariesXudong Wang, Ying Zhu, Qingyi Zhao, et al.ACS Medicinal Chemistry Letters|April 17, 2024
Empowering Voices: Inspiring Women in Medicinal ChemistryMaria-Jesus Blanco, Joanne J Bronson, Erin F DiMauro, et al.ACS Medicinal Chemistry Letters|January 14, 2026
Controlling Temozolomide Efficacy by Light-Dependent Inhibition of O6‑Methylguanine DNA MethyltransferaseIvonne R Lopez-Miranda, Josef I Sim, Gabrielle Juneau, et al.ACS Medicinal Chemistry Letters|January 14, 2026
Selective TYK2 Inhibition, Prenatal Cell Diagnostics, and Biomarker-Guided Immunotherapy: Expanding Precision MedicineMahmoud A Elkhalifa, Robert B KargboACS Medicinal Chemistry Letters|January 14, 2026
Synthesis and Evaluation of a 99mTc-Labeled Fibroblast Activation Protein (FAP)-Specific Radiotracer for SPECT ImagingTianhong Yang, Lingyu Xue, Lei Peng, et al.ACS Medicinal Chemistry Letters|January 14, 2026
A Novel Class of Orally Bioavailable Phenylglycine-Benzoxaborole Conjugates with Antimalarial Activity and Potentially Novel Mechanism of ActionMokhitli Morake, Dale Taylor, Dina Coertzen, et al.Pageof 441