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ACS Medicinal Chemistry Letters|July 19, 2023
The Quest for Oral PROTAC drugs: Evaluating the Weaknesses of the Screening PipelineGiulia Apprato, Giuseppe Ermondi, Giulia CaronACS Medicinal Chemistry Letters|July 19, 2023
Discovery of Potent, Dual-Inhibitors of Diacylglycerol Kinases Alpha and Zeta Guided by Phenotypic OptimizationLouis Chupak, Michael Wichroski, Xiaofan Zheng, et al.ACS Medicinal Chemistry Letters|July 19, 2023
Microbiome-Gut-Brain Axis Modulation: New Approaches in Treatment of Parkinson's Disease and Amyotrophic Lateral SclerosisRobert B KargboACS Medicinal Chemistry Letters|July 19, 2023
Examination of the Impact of Triazole Position within Linkers on Solubility and Lipophilicity of a CDK9 Degrader SeriesOluwatosin R Ayinde, Chia Sharpe, Emily Stahl, et al.ACS Medicinal Chemistry Letters|July 19, 2023
Unveiling New KRASG12D Inhibitors: A Promising Approach for Pancreatic Cancer TherapyRobert B KargboACS Medicinal Chemistry Letters|August 16, 2023
Structure-Activity Relationship Study of 1H-Pyrrole-3-carbonitrile Derivatives as STING Receptor AgonistsChang Shen, Peijia Xu, Changfa Zhang, et al.ACS Medicinal Chemistry Letters|August 16, 2023
Pyridazine Derivatives as NLRP3 Inhibitors for Treating Asthma, COPD, Parkinson's Disease, and Alzheimer's DiseaseRam W SabnisACS Medicinal Chemistry Letters|August 16, 2023
Design, Construction, and Screening of Diversified Pyrimidine-Focused DNA-Encoded LibrariesMengnisa Seydimemet, Yixuan Yang, Yuhan Lv, et al.ACS Medicinal Chemistry Letters|August 16, 2023
Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric ModulatorMichael T Rudd, Peter J Manley, Barbara Hanney, et al.ACS Medicinal Chemistry Letters|August 16, 2023
The Synergistic Effects of 5-HT2A and TRP Agonism/Antagonism in Reducing Inflammation for Enhanced Mental and Physical HealthRobert B KargboPageof 441