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ACS Medicinal Chemistry Letters|April 16, 2025
Novel Piperidinylpyridinylcarbonitrile Derivatives as QPCT and QPCTL Inhibitors for Treating CancerRam W SabnisACS Medicinal Chemistry Letters|June 18, 2025
Triazine Macrocycle Libraries: Synthesis, logD Prediction, and a Surprisingly Hydrophobic, Membrane-Permeable DiamineGretel A Stokes, Casey J Patterson-Gardner, Alexander M Engstrom, et al.ACS Medicinal Chemistry Letters|June 18, 2025
FAK: A Potential Target for Cancer TherapyChao Zhang, Yu RaoACS Medicinal Chemistry Letters|June 18, 2025
SSTR-Mediated Precision Delivery: Overcoming Triptolide's Limitations through Octreotide Conjugation in Pancreatic Cancer TreatmentDandan Su, Qiaohong Bao, Xinyu Wang, et al.ACS Medicinal Chemistry Letters|June 18, 2025
Novel Tetrahydrocyclohepteneindole Derivatives Targeting Estrogen Receptor Alpha for the Treatment of Breast CancerZhendong Song, Steven H LiangACS Medicinal Chemistry Letters|June 18, 2025
Novel Indole Derivatives as Serotonergic Psychedelic Agents for Treating Psychosis, Mental Illness, and CNS DisordersRam W SabnisACS Medicinal Chemistry Letters|June 18, 2025
Discovery of Reversible, Noncovalent Bruton's Tyrosine Kinase Inhibitors Targeting BTK C481S MutationDebasis Das, Lingzhi Xie, Dandan Qiao, et al.ACS Medicinal Chemistry Letters|May 14, 2025
Novel Tetrahydrobenzo[b]pyrazolo[3,4-e][1,4]diazepine Compounds as Oxytocin Receptor Agonists for Treating Autism Spectrum DisordersZhendong Song, Steven H LiangACS Medicinal Chemistry Letters|May 14, 2025
Targeting KRAS G12D Mutations: Advances in Small Molecule Inhibitors and PROTAC TechnologyRobert B KargboACS Medicinal Chemistry Letters|May 14, 2025
Gold(I) N-Heterocyclic Carbene Complexes as Ferroptosis Inducing Anticancer AgentsEvelyn Schlegel, Zisis Papadopoulos, Nicolás Montesdeoca, et al.Pageof 441