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ACS Medicinal Chemistry Letters|August 20, 2025
Novel Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitors for the Treatment of Parkinson's DiseaseZhendong Song, Steven H LiangACS Medicinal Chemistry Letters|August 20, 2025
Novel Tricyclic Triazolo Compounds as DGK Inhibitors for Treating Metastatic MelanomaRam W SabnisACS Medicinal Chemistry Letters|August 20, 2025
Novel Peptides as GIPR/GLP-1R/GCGR Triagonists for Treating Type 2 Diabetes MellitusQilong Hu, Steven H LiangACS Medicinal Chemistry Letters|August 20, 2025
Novel Azepinoindoles as 5‑HT2C Agonists for Treating Depression, Drug Addiction, Alcoholism, PTSD, and Neuropathic PainRam W SabnisACS Medicinal Chemistry Letters|August 20, 2025
Novel 3‑(2-(Aminoethyl)-indol-4-ol Derivatives as 5‑HT2C Agonists for Treating Depression, Alcoholism, Drug Addiction, PTSD, and Seizure DisordersRam W SabnisACS Medicinal Chemistry Letters|August 20, 2025
Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water MoleculeMark E Schnute, Gary M Chinigo, Kentaro Futatsugi, et al.ACS Medicinal Chemistry Letters|August 22, 2025
2‑Aminoimidazole-benzimidazole Conjugates Potentiate the Gram-Positive Selective Antibiotic Clarithromycin against Acinetobacter baumanniiAshley N Crotteau, Ansley M Nemeth, Roberta J Melander, et al.ACS Medicinal Chemistry Letters|February 12, 2026
Discovery of N-Acetyltransferase 8-Like (NAT8L) inhibitors based on a N-Acylated (Piperidin-3-ylmethyl)-1,2,4-Oxadiazole ScaffoldMd Junayed Nayeen, Ajit G Thomas, Biswajit Kundu, et al.ACS Medicinal Chemistry Letters|March 19, 2025
Enhanced Cytotoxicity of [10]-Gingerol-Coumarin-Triazole Hybrid as a Theranostic Agent for Triple Negative Breast CancerArthur Deponte Zutião, Bianca Cruz Pachane, Paulo Sérgio Gonçalves Nunes, et al.ACS Medicinal Chemistry Letters|March 19, 2025
Novel Piperazine Derivatives as Selective Antagonists of GluN2B-Containing NMDARs under Acidic pH ConditionsYinlong Li, Steven H LiangPageof 441