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ACS Medicinal Chemistry Letters|March 16, 2018
Potential Antimicrobial Isopropanol-Conjugated Carbazole Azoles as Dual Targeting Inhibitors of Enterococcus faecalisYuan Zhang, Vijai Kumar Reddy Tangadanchu, Yu Cheng, et al.
ACS Medicinal Chemistry Letters|March 16, 2018
Y08060: A Selective BET Inhibitor for Treatment of Prostate CancerQiuping Xiang, Yan Zhang, Jiaguo Li, et al.
ACS Medicinal Chemistry Letters|March 16, 2018
Elimination of HIV-1 Latently Infected Cells by Gnidimacrin and a Selective HDAC InhibitorLi Huang, Wei-Hong Lai, Lei Zhu, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
3,5-Disubstituted-indole-7-carboxamides as IKKβ Inhibitors: Optimization of Oral Activity via the C3 SubstituentJeffrey K Kerns, Jakob Busch-Petersen, Wei Fu, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)Jun Li, Lawrence J Kennedy, Steven J Walker, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
Privileged Structures and Polypharmacology within and between Protein FamiliesJoshua Meyers, Nicola E A Chessum, Salyha Ali, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
Structure-Property Basis for Solving Transporter-Mediated Efflux and Pan-Genotypic Inhibition in HCV NS5B InhibitorsKap-Sun Yeung, Brett R Beno, Kathy Mosure, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
Modification of the Thioglycosyl-Naphthalimides as Potent and Selective Human O-GlcNAcase InhibitorsShengqiang Shen, Lili Dong, Wei Chen, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
In Vitro Ligand Binding Kinetics Explains the Pharmacokinetics of [18F]FE-PE2I in Dopamine Transporter PET ImagingSiim Kukk, Olavi Loog, Jukka-Veli Hiltunen, et al.
ACS Medicinal Chemistry Letters|January 8, 2019
Novel Fluorescence Competition Assay for Retinoic Acid Binding ProteinsCharles W E Tomlinson, David R Chisholm, Roy Valentine, et al.
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