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ACS Medicinal Chemistry Letters|November 22, 2019
Discovery of Pyrazolocarboxamides as Potent and Selective Receptor Interacting Protein 2 (RIP2) Kinase InhibitorsCurt D Haffner, Adam K Charnley, Christopher J Aquino, et al.ACS Medicinal Chemistry Letters|November 22, 2019
Scaffold Morphing Identifies 3-Pyridyl Azetidine Ureas as Inhibitors of Nicotinamide Phosphoribosyltransferase (NAMPT)Daniel S Palacios, Erik L Meredith, Toshio Kawanami, et al.ACS Medicinal Chemistry Letters|November 22, 2019
INCB050465 (Parsaclisib), a Novel Next-Generation Inhibitor of Phosphoinositide 3-Kinase Delta (PI3Kδ)Eddy W Yue, Yun-Long Li, Brent Douty, et al.ACS Medicinal Chemistry Letters|December 22, 2017
Correction to "Apratoxin S10, a Dual Inhibitor of Angiogenesis and Cancer Cell Growth To Treat Highly Vascularized Tumors"Weijing Cai, Qi-Yin Chen, Long H Dang, et al.ACS Medicinal Chemistry Letters|December 21, 2017
Synthesis of Novel Selenides Bearing Benzenesulfonamide Moieties as Carbonic Anhydrase I, II, IV, VII, and IX InhibitorsAndrea Angeli, Damiano Tanini, Antonella Capperucci, et al.ACS Medicinal Chemistry Letters|December 21, 2017
EGFR-Targeted Magnetic Nanovectors Recognize, in Vivo, Head and Neck Squamous Cells Carcinoma-Derived TumorsDavid Colecchia, Elena Nicolato, Costanza Ravagli, et al.ACS Medicinal Chemistry Letters|December 21, 2017
2-Arylidene Hydrazinecarbodithioates as Potent, Selective Inhibitors of Cystathionine γ-Lyase (CSE)Abir Bhattacharjee, Antara Sinha, Kiira Ratia, et al.ACS Medicinal Chemistry Letters|December 21, 2017
Synthesis and Evaluation of Radiolabeled Phosphoramide Mustard with Selectivity for Hypoxic Cancer CellsWenting Zhang, Wei Fan, Zhengyuan Zhou, et al.ACS Medicinal Chemistry Letters|December 21, 2017
Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous BasesAlessio Nocentini, Silvia Bua, Carrie L Lomelino, et al.ACS Medicinal Chemistry Letters|December 21, 2017
VU6010608, a Novel mGlu7 NAM from a Series of N-(2-(1H-1,2,4-Triazol-1-yl)-5-(trifluoromethoxy)phenyl)benzamidesCarson W Reed, Kevin M McGowan, Paul K Spearing, et al.Pageof 441