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ACS Medicinal Chemistry Letters|May 22, 2020
Synthetic Sphingolipids with 1,2-Pyridazine Appendages Improve Antiproliferative Activity in Human Cancer Cell LinesSylvestre P J T Bachollet, Vito Vece, Alison N McCracken, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Synthesis, Antiproliferative Effect, and Topoisomerase II Inhibitory Activity of 3-Methyl-2-phenyl-1H-indolesNace Zidar, Daniela Secci, Tihomir Tomašič, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Glycomimetic Based Approach toward Selective Carbonic Anhydrase InhibitorsDebora Pratesi, Camilla Matassini, Andrea Goti, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Structural Elucidation and Antimicrobial Characterization of Novel Diterpenoids from Fabiana densa var. ramulosaDeborah Quaglio, Silvia Corradi, Silvia Erazo, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Peptides Mimicking the β7/β8 Loop of HIV-1 Reverse Transcriptase p51 as "Hotspot-Targeted" Dimerization InhibitorsPedro A Sánchez-Murcia, Sonia de Castro, Carlos García-Aparicio, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE InhibitorMarco Catto, Leonardo Pisani, Eugenio de la Mora, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
BOPC1 Enantiomers Preparation and HuR Interaction Study. From Molecular Modeling to a Curious DEEP-STD NMR ApplicationSerena Della Volpe, Roberta Listro, Michela Parafioriti, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Design of First-in-Class Dual EZH2/HDAC Inhibitor: Biochemical Activity and Biological Evaluation in Cancer CellsAnnalisa Romanelli, Giulia Stazi, Rossella Fioravanti, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
Substituted Naphthalenediimide Compounds Bind Selectively to Two Human Quadruplex Structures with Parallel TopologyTam Vo, Sally Oxenford, Richard Angell, et al.
ACS Medicinal Chemistry Letters|May 22, 2020
HOPPI-NMR: Hot-Peptide-Based Screening Assay for Inhibitors of Protein-Protein Interactions by NMRDiego Brancaccio, Salvatore Di Maro, Linda Cerofolini, et al.
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