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ACS Medicinal Chemistry Letters|April 15, 2026
Synthesis and LCMS Characterization of a 1275-Member Library of 24-Atom Triazine Macrocycles Derived from Quantitative Dimerization Occurring with >99.9% FidelityLiam E Claton, K Harsha Vardan Reddy, Samantha N Gaines, et al.ACS Medicinal Chemistry Letters|April 15, 2026
Discovery and Optimization of a Trichloroacetamidine Scaffold as a Novel Antibacterial against Multidrug-Resistant Staphylococcus aureusLeticia Christina Pires Gonçalves, Zakaria Moutaoukil, Juan A Garcia-Sanchez, et al.ACS Medicinal Chemistry Letters|April 15, 2026
SAR-Guided Scaffold Innovation of Selective V2R Antagonists: Therapeutic Frontiers in ADPKDHaofeng Shi, Yinlong Li, Steven H LiangACS Medicinal Chemistry Letters|April 15, 2026
Potent Neuronal Nicotinamide Adenine Dinucleotide-Boosting Tetrahydroquinoxalines: Structure-Activity Relationships and Early Drug Metabolism and Pharmacokinetics EvaluationPetra Cuřínová, Melissa Jöe, Filip Cesar, et al.ACS Medicinal Chemistry Letters|April 15, 2026
BBB-Permeable PROTACs: Where Do We Stand?Serena Francisco, Giulia Apprato, Matteo Rossi Sebastiano, et al.ACS Medicinal Chemistry Letters|March 18, 2026
Emerging Paradigms in Immune-Focused Drug DiscoveryAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|March 18, 2026
Discovery of Pan-TEAD Inhibitors That Disrupt YAP-TEAD Interaction as a Potential Therapy for Gastric Cancers and Mutant KRAS and EGFR Lung CancersRamesh Kumar, Joanne Thian, Joel D W Toh, et al.ACS Medicinal Chemistry Letters|March 18, 2026
Modulation of Cancer Networks through Protein Degradation, DNA Repair Inhibition, and Quantitative InteractomicsAnna C Renner, Robert B KargboACS Medicinal Chemistry Letters|March 18, 2026
Synthesis of Novel STING Antagonists and Their Uses in Treatment of STING Related DiseasesHaofeng Shi, Steven H LiangACS Medicinal Chemistry Letters|March 18, 2026
6,7-Dihalo-Benzothiadiazines as Potent and Selective AMPA Receptor Modulators for Cognitive Enhancement and NeuroprotectionYinlong Li, Hongjie Yuan, Steven H LiangPageof 438