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ACS Medicinal Chemistry Letters|July 21, 2022
Discovery and Optimization of Seven-Membered Lactam-Based Compounds to Phenocopy the Inhibition of the Aurora Kinase BJian Huang, Qiong Shi, Namrta Choudhry, et al.ACS Medicinal Chemistry Letters|July 21, 2022
Indolactam Dipeptides as Nanomolar Gli InhibitorsManuel Mendoza, UyenPhuong Tran, Grace C Zhang, et al.ACS Medicinal Chemistry Letters|July 21, 2022
Discovery of Antibacterial Contezolid Acefosamil: Innovative O-Acyl Phosphoramidate Prodrug for IV and Oral TherapiesJinqian Liu, Wen Wang, Changqing Wang, et al.ACS Medicinal Chemistry Letters|July 21, 2022
Discovery of Novel Pyrazolopyrimidines as Potent, Selective, and Orally Bioavailable Inhibitors of ALK2Minh H Nguyen, Onur Atasoylu, Liangxing Wu, et al.ACS Medicinal Chemistry Letters|May 17, 2023
Quantum Annealing Designs Nonhemolytic Antimicrobial Peptides in a Discrete Latent SpaceAndrejs Tučs, Francois Berenger, Akiko Yumoto, et al.ACS Medicinal Chemistry Letters|May 17, 2023
Synthesis of Artesunic Acid-Coumarin Hybrids as Potential Antimelanoma AgentsClaudio Zippilli, Silvia Filippi, Silvia Cesarini, et al.ACS Medicinal Chemistry Letters|May 17, 2023
PROTAC: Harnessing Targeted Chimeras for Selective BCL-2 Degradation in Cancer TreatmentRobert B KargboACS Medicinal Chemistry Letters|May 17, 2023
Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant CompoundsAntonella Ilenia Alfano, Sveva Pelliccia, Giacomo Rossino, et al.ACS Medicinal Chemistry Letters|May 17, 2023
Addressing the Osimertinib Resistance Mutation EGFR-L858R/C797S with Reversible AminopyrimidinesTobias Grabe, Kirujan Jeyakumar, Janina Niggenaber, et al.Pageof 438