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ACS Pharmacology & Translational Science|July 29, 2025
Oral Prodrug of a Novel Glutathione Surrogate Reverses Metabolic Dysregulation and Attenuates Neurodegenerative Process in Transgenic Alzheimer's MiceSwetha Pavani Rao, Aminat O Imam-Fulani, Wei Xie, et al.ACS Pharmacology & Translational Science|August 4, 2025
Limosilactobacillus fermentum M5e Attenuates Hyperuricemia and Renal Injury via Dual Modulation of Gut Microbiota and Purine Metabolic PathwaysYi He, Dilinuer Aikepa, Meiting Liang, et al.ACS Pharmacology & Translational Science|January 18, 2023
Detailed Insights into the Inhibitory Mechanism of New Ebselen Derivatives against Main Protease (Mpro) of Severe Acute Respiratory Syndrome Coronavirus-2 (SARS-CoV-2)Pritiranjan Sahoo, Dipti Ranjan Lenka, Monojit Batabyal, et al.ACS Pharmacology & Translational Science|January 19, 2023
Behavioral and Proteomic Studies Reveal Methylglyoxal Activate Pathways Associated with Alzheimer's DiseaseGouri Patil, Shabda Kulsange, Rubina Kazi, et al.ACS Pharmacology & Translational Science|January 19, 2023
Inhibition of Protein Disulfide Isomerase (PDIA1) Leads to Proteasome-Mediated Degradation of Ubiquitin-like PHD and RING Finger Domain-Containing Protein 1 (UHRF1) and Increased Sensitivity of Glioblastoma Cells to Topoisomerase II InhibitorsRima Mouawad, Nouri NeamatiACS Pharmacology & Translational Science|January 19, 2023
Cell-Permeable PROTAC Degraders against KEAP1 Efficiently Suppress Hepatic Stellate Cell Activation through the Antioxidant and Anti-Inflammatory PathwayFengqin Wang, Ying Zhan, Manman Li, et al.ACS Pharmacology & Translational Science|June 21, 2021
Dual-Targeting and Stimuli-Triggered Liposomal Drug Delivery in Cancer TreatmentNour AlSawaftah, William G Pitt, Ghaleb A HusseiniACS Pharmacology & Translational Science|June 21, 2021
Selective Targeting of Vascular Endothelial YAP Activity Blocks EndMT and Ameliorates Unilateral Ureteral Obstruction-Induced Kidney FibrosisYafeng Ren, Yuwei Zhang, Lu Wang, et al.ACS Pharmacology & Translational Science|June 21, 2021
Inhibition of Histone Deacetylases 1, 2, and 3 Enhances Clearance of Cholesterol Accumulation in Niemann-Pick C1 FibroblastsDana L Cruz, Nina Pipalia, Shu Mao, et al.ACS Pharmacology & Translational Science|June 21, 2021
Discovery of μ,δ-Opioid Receptor Dual-Biased Agonists That Overcome the Limitation of Prior Biased AgonistsJin Hee Lee, Suh-Youn Shon, Woojin Jeon, et al.Pageof 139