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ACS Pharmacology & Translational Science|January 15, 2026
3‑(4-Hydroxyphenyl-1,2,3-Triazol-1-yl)Quinuclidine, a Selective α7 Nicotinic Acetylcholine Receptor Agonist, Attenuates Inflammatory Pain with a Favorable Central Nervous System Safety Profile in MiceThorsang Weerakul, Hasriadi, Krittamate Chatdamrongsakool, et al.ACS Pharmacology & Translational Science|January 15, 2026
Structural Pharmacology of Estrogen-Related ReceptorsPuhan Zhao, Hong Fang, Bahaa Elgendy, et al.ACS Pharmacology & Translational Science|January 15, 2026
Potent Competitive Inhibitors of Ecto-5'-nucleotidase (CD73) based on 6‑(Het)aryl-7-deazapurine Ribonucleoside 5'‑O‑BisphosphonatesUgnė Šinkevičiu̅tė, Magdalena Šímová, Radek Staník, et al.ACS Pharmacology & Translational Science|January 15, 2026
Optimization of a Green Extraction Technique for Kratom (Ketum) Leaf Extract via Accelerated Solvent Extraction: Phytochemical Profiles, Cytotoxicity, and Antinociceptive ActivityNurul Najwa Rusmadi, Thiruventhan Karunakaran, Faiqah Ramli, et al.ACS Pharmacology & Translational Science|January 15, 2026
Protease-Activated Receptor 4 (PAR4)-Tethered Ligand Antagonists Demonstrate Thrombin LiabilityEmma M Webb, Jackson B Cassada, Heidi E HammACS Pharmacology & Translational Science|January 15, 2026
Neuronal Organoid Engineering and Disease-Focused High-Throughput Neuropharmacology: Advances, Limitations, and Translational StrategiesBahareh Farasati Far, Kimia Omidvar, Ehsan Heidari, et al.ACS Pharmacology & Translational Science|November 20, 2025
Crescent-Shaped Xanthone-Benzimidazole Conjugates as New Target Probes for Telomeric G‑Quadruplex DNA and Specific Cytotoxicity on Cancer CellsPulakesh Pramanik, Bappa Maiti, Santanu BhattacharyaACS Pharmacology & Translational Science|November 20, 2025
Conformational Heterogeneity Underlying Divergent Signaling in Class A G Protein-Coupled ReceptorsKyriakos Georgiou, Antonios KolocourisACS Pharmacology & Translational Science|November 20, 2025
Development and Preclinical Evaluation of a Zirconium-89-Labeled Immunoconjugate for Positron Emission Tomography Imaging of Leukemia Inhibitory Factor in GlioblastomaEmily Betancourt Fernández, Julia Baguña Torres, Raffaella Iurlaro, et al.ACS Pharmacology & Translational Science|November 20, 2025
Lands' Cycle at the Crossroads: Phospholipid Remodelling, Oxidative Stress, Cellular Toxicity, and Therapeutic TargetingAiram Roggero, Marcos H Toyama, Sergio F SousaPageof 139