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Acta Pharmacologica Sinica|August 21, 2025
ALKBH5 deficiency suppresses hepatocarcinogenesis in mice via m6A-dependent STAT1 restorationKai-Ting Wang, Shuai Yang, Zi-Han Zhao, et al.Acta Pharmacologica Sinica|February 6, 2026
CSF1R inhibitor C19 for glioma immunotherapy enabled by brain-targeting liposomal deliveryWen-Qin Song, Yue-Qian Wu, Quan-Feng Zhu, et al.Acta Pharmacologica Sinica|February 3, 2026
Chronic 5-HT7R activation drives depressive phenotypes and synaptic dysfunctionBartłomiej Pochwat, Julia Masternak, Bartosz Bobula, et al.Acta Pharmacologica Sinica|January 29, 2026
A structural overview of G-protein-coupled receptors in neurological disordersOindrilla Dutta Gupta, Indranil Chakraborty, Kuntal PalActa Pharmacologica Sinica|February 6, 2026
PDE4 inhibitor rolipram dynamically regulates the balance between D1-MSNs and D2-MSNs in the DMS to modulate abnormal "Go" behavior associated with alcohol addictionWei Zhao, Shuang Zhao, Zi-Qi Wang, et al.Acta Pharmacologica Sinica|January 27, 2026
ER-phagy receptors: structural mechanisms in selective ER degradation and disease implicationsWen-Jing Yang, Rui ShengActa Pharmacologica Sinica|January 20, 2026
A novel photosensitizer berberine derivative B12 induces apoptosis and suppresses HIF-1α expression in colorectal cancer cells via mitochondria-to-nucleus sequential-targetingWen-Bin Pei, Zi-Yu Lei, Fu-Quan Xie, et al.Acta Pharmacologica Sinica|March 21, 2025
Microemulsion-based drug delivery system identifies pepper alkaloids as anti-obesity compoundsTian-Kai Meng, Ruo-Lei Han, Peng Ma, et al.Acta Pharmacologica Sinica|March 22, 2025
Anti-EGFR therapy can overcome acquired resistance to the third-generation ALK-tyrosine kinase inhibitor lorlatinib mediated by activation of EGFRChen Hu, Cong-Hua Lu, Jie Zheng, et al.Acta Pharmacologica Sinica|March 18, 2025
Transport mechanism and drug discovery of human monocarboxylate transporter 1Sai Shi, Jia-Chen Li, Xiao-Yu Zhou, et al.Pageof 545