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Bioorganic & Medicinal Chemistry|November 29, 2021
Novel O-acylated (E)-3-aryl-6,7-dihydrobenzisoxazol-4(5H)-one oximes targeting HSP90-HER2 axis in breast cancer cellsYuri A Piven, Margarita A Yastrebova, Alvina I Khamidullina, et al.
Bioorganic & Medicinal Chemistry|November 21, 2018
Synthesis and biological evaluation of thielocin B1 analogues as protein-protein interaction inhibitors of PAC3 homodimerKosuke Ohsawa, Masahito Yoshida, Miho Izumikawa, et al.
Bioorganic & Medicinal Chemistry|February 17, 2019
Structure-based virtual screening for insect ecdysone receptor ligands using MM/PBSAShinri Horoiwa, Taiyo Yokoi, Satoru Masumoto, et al.
Bioorganic & Medicinal Chemistry|February 19, 2019
Design, synthesis and biological evaluation of inhibitors of cathepsin K on dedifferentiated chondrocytesXiao-Yu Yuan, Zhongyuan Ren, Yuqing Wu, et al.
Bioorganic & Medicinal Chemistry|February 19, 2019
4,6-Substituted-1H-Indazoles as potent IDO1/TDO dual inhibitorsLingling Yang, Yang Chen, Junlin He, et al.
Bioorganic & Medicinal Chemistry|February 19, 2019
Anti-cancer activity of m-carborane-containing trimethoxyphenyl derivatives through tubulin polymerization inhibitionAsako Kaise, Yasuyuki Endo, Kiminori Ohta
Bioorganic & Medicinal Chemistry|February 20, 2019
Design and synthesis of potent myostatin inhibitory cyclic peptidesCédric Rentier, Kentaro Takayama, Mariko Saitoh, et al.
Bioorganic & Medicinal Chemistry|March 9, 2019
Synthesis and radical-scavenging activity of C-methylated fisetin analoguesKohei Imai, Ikuo Nakanishi, Kei Ohkubo, et al.
Bioorganic & Medicinal Chemistry|March 10, 2019
Inhibition of the FAD containing ER oxidoreductin 1 (Ero1) protein by EN-460 as a strategy for treatment of multiple myelomaKaren E Hayes, Paratchata Batsomboon, Wei-Chih Chen, et al.
Bioorganic & Medicinal Chemistry|March 10, 2019
Structural requirement of tunicamycin V for MraY inhibitionKazuki Yamamoto, Akira Katsuyama, Satoshi Ichikawa
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