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Bioorganic & Medicinal Chemistry|January 31, 2021
Insights into non-peptide small-molecule inhibitors of the PD-1/PD-L1 interaction: Development and perspectiveXia Wu, Yangyang Meng, Lei Liu, et al.Bioorganic & Medicinal Chemistry|February 1, 2021
Quest for a potent antimalarial drug lead: Synthesis and evaluation of 6,7-dimethoxyquinazoline-2,4-diaminesYuki Mizukawa, Mayumi Ikegami-Kawai, Masako Horiuchi, et al.Bioorganic & Medicinal Chemistry|January 30, 2021
Potential inhibitors interacting in Neuropilin-1 to develop an adjuvant drug against COVID-19, by molecular dockingJosé Luis Vique-SánchezBioorganic & Medicinal Chemistry|January 19, 2021
Synthesis, anticancer activity and molecular docking studies of N-deacetylthiocolchicine and 4-iodo-N-deacetylthiocolchicine derivativesGreta Klejborowska, Alicja Urbaniak, Ewa Maj, et al.Bioorganic & Medicinal Chemistry|January 21, 2021
Design, synthesis and biological evaluation of novel indanone containing spiroisoxazoline derivatives with selective COX-2 inhibition as anticancer agentsHoda Abolhasani, Afshin Zarghi, Tahereh Komeili Movahhed, et al.Bioorganic & Medicinal Chemistry|February 7, 2021
Discovery of benzo[f]pyrido[4,3-b][1,4]oxazepin-10-one derivatives as orally available bromodomain and extra-terminal domain (BET) inhibitors with efficacy in an in vivo psoriatic animal modelMasanori Sato, Takekazu Kondo, Yasushi Kohno, et al.Bioorganic & Medicinal Chemistry|January 13, 2021
Novel arylcarbamate-N-acylhydrazones derivatives as promising BuChE inhibitors: Design, synthesis, molecular modeling and biological evaluationDiego A S Yamazaki, Andrew M F Rozada, Paula Baréa, et al.Bioorganic & Medicinal Chemistry|January 13, 2021
1,2,4-Thiadiazole acyclic nucleoside phosphonates as inhibitors of cysteine dependent enzymes cathepsin K and GSK-3βAlice Pomeislová, Miroslav Otmar, Petra Rubešová, et al.Bioorganic & Medicinal Chemistry|January 14, 2021
A comprehensive review on the biological interest of quinoline and its derivativesBasavarajaiah Suliphuldevara Matada, Raviraj Pattanashettar, Nagesh Gunavanthrao YernaleBioorganic & Medicinal Chemistry|July 30, 2019
Synthesis and evaluation of novel potent TSPO PET ligands with 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamideVan Hieu Tran, Hyunjun Park, Jaekyung Park, et al.Pageof 1,701