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Bioorganic & Medicinal Chemistry|January 3, 2022
Berberine improves liver injury induced glucose and lipid metabolic disorders via alleviating ER stress of hepatocytes and modulating gut microbiota in miceLanxiang Yang, Siping Yu, Yanhong Yang, et al.Bioorganic & Medicinal Chemistry|January 16, 2022
Development of a radioiodinated thioflavin-T-Congo-red hybrid probe for diagnosis of systemic amyloidosisYoshie Haratake, Kohei Sano, Miki Tsuchiya, et al.Bioorganic & Medicinal Chemistry|January 7, 2022
Indole derivatives as tubulin polymerization inhibitors for the development of promising anticancer agentsYu Hong, Yuan-Yuan Zhu, Qiuqin He, et al.Bioorganic & Medicinal Chemistry|January 9, 2022
Oligonucleotides containing 2'-O-methyl-5-(1-phenyl-1,2,3-triazol-4-yl)uridines demonstrate increased affinity for RNA and induce exon-skipping in vitroAlejandro Gimenez Molina, Prithi Raguraman, Line Delcomyn, et al.Bioorganic & Medicinal Chemistry|December 31, 2021
Synthesis of sorbicillinoid analogues with anti-inflammation activitiesMeng Zhang, Fangfang Wang, Wenjuan Ding, et al.Bioorganic & Medicinal Chemistry|January 20, 2022
Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding ActivityFumie Sakurai, Takafumi Yukawa, Asato Kina, et al.Bioorganic & Medicinal Chemistry|January 20, 2022
Directly arylated oligonucleotides as fluorescent molecular rotors for probing DNA single-nucleotide polymorphismsGuralamatta Siddappa Ravi Kumara, Young Jun SeoBioorganic & Medicinal Chemistry|May 6, 2008
Muscarinic antagonists with multiple stereocenters: Synthesis, affinity profile and functional activity of isomeric 1-methyl-2-(2,2-alkylaryl-1,3-oxathiolan-5-yl)pyrrolidine sulfoxide derivativesSilvia Dei, Cristina Bellucci, Michela Buccioni, et al.Bioorganic & Medicinal Chemistry|May 7, 2008
Anti-Helicobacter pylori activity of derivatives of the phthalide-containing antibacterial agents spirolaxine methyl ether, CJ-12,954, CJ-13,013, CJ-13,102, CJ-13,104, CJ-13,108 and CJ-13,015Fiona J Radcliff, John D Fraser, Zoe E Wilson, et al.Bioorganic & Medicinal Chemistry|April 18, 2008
Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 6: Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocineMark P Wentland, Xufeng Sun, Dana J Cohen, et al.Pageof 1,701