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Bioorganic & Medicinal Chemistry|May 11, 2011
Quinoline-4-methyl esters as human nonpancreatic secretory phospholipase A₂ inhibitorsYiran Wu, Zheng Chen, Ying Liu, et al.Bioorganic & Medicinal Chemistry|May 4, 2011
Design and evaluation of 3-aminopyrazolopyridinone kinase inhibitors inspired by the natural product indirubinLynette A Smyth, Thomas P Matthews, Ian CollinsBioorganic & Medicinal Chemistry|March 29, 2011
Acyl derivatives of p-aminosulfonamides and dapsone as new inhibitors of the arginine methyltransferase hPRMT1Elisabeth-Maria Bissinger, Ralf Heinke, Astrid Spannhoff, et al.Bioorganic & Medicinal Chemistry|March 29, 2011
Inhibitory effects of Mannich bases of heterocyclic chalcones on NO production by activated RAW 264.7 macrophages and superoxide anion generation and elastase release by activated human neutrophilsM Vijaya Bhaskar Reddy, Tsong-Long Hwang, Yann-Lii Leu, et al.Bioorganic & Medicinal Chemistry|April 29, 2011
Thiazole-based chalcones as potent antimicrobial agents. Synthesis and biological evaluationK Liaras, A Geronikaki, J Glamočlija, et al.Bioorganic & Medicinal Chemistry|April 29, 2011
Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR4Ryo Masuda, Shinya Oishi, Hiroaki Ohno, et al.Bioorganic & Medicinal Chemistry|April 29, 2011
Avoidance of the Ames test liability for aryl-amines via computationPatrick McCarren, Gregory R Bebernitz, Peter Gedeck, et al.Bioorganic & Medicinal Chemistry|April 15, 2011
Evaluation of superior BACE1 cleavage sequences containing unnatural amino acidsTaeko Kakizawa, Akira Sanjoh, Akane Kobayashi, et al.Bioorganic & Medicinal Chemistry|June 11, 2011
Discovery of 4-[4-({(3R)-1-butyl-3-[(R)-cyclohexyl(hydroxy)methyl]-2,5-dioxo-1,4,9-triazaspiro[5.5]undec-9-yl}methyl)phenoxy]benzoic acid hydrochloride: a highly potent orally available CCR5 selective antagonistRena Nishizawa, Toshihiko Nishiyama, Katsuya Hisaichi, et al.Bioorganic & Medicinal Chemistry|November 9, 2011
Capturing of the free cysteine residue in the ligand-binding site by affinity labeling of the ORL1 nociceptin receptorAyami Matsushima, Hirokazu Nishimura, Shogo Inamine, et al.Pageof 1,701