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Bioorganic & Medicinal Chemistry|October 12, 2010
Structure-activity relationships for inhibition of inosine monophosphate dehydrogenase and differentiation induction of K562 cells among the mycophenolic acid derivativesShinya Mitsuhashi, Junichi Takenaka, Katsushige Iwamori, et al.Bioorganic & Medicinal Chemistry|October 12, 2010
Design, synthesis and bioevaluation of dihydropyrazolo[3,4-b]pyridine and benzo[4,5]imidazo[1,2-a]pyrimidine compounds as dual KSP and Aurora-A kinase inhibitors for anti-cancer agentsRong-Geng Fu, Qi-Dong You, Lei Yang, et al.Bioorganic & Medicinal Chemistry|October 13, 2010
Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligandsMaria Paola Giovannoni, Claudia Vergelli, Agostino Cilibrizzi, et al.Bioorganic & Medicinal Chemistry|September 9, 2010
OGA inhibition by GlcNAc-selenazolineEun Ju Kim, Dona C Love, Etzer Darout, et al.Bioorganic & Medicinal Chemistry|October 8, 2010
Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIIIEdita Čapkauskaitė, Lina Baranauskienė, Dmitrij Golovenko, et al.Bioorganic & Medicinal Chemistry|February 18, 2011
Cofactor-type inhibitors of inosine monophosphate dehydrogenase via modular approach: targeting the pyrophosphate binding sub-domainKrzysztof Felczak, Liqiang Chen, Daniel Wilson, et al.Bioorganic & Medicinal Chemistry|February 26, 2011
CD22-antagonists with nanomolar potency: the synergistic effect of hydrophobic groups at C-2 and C-9 of sialic acid scaffoldHajjaj H M Abdu-Allah, Kozo Watanabe, Gladys C Completo, et al.Bioorganic & Medicinal Chemistry|March 1, 2011
Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitorsSilviya D Furdas, Suhaib Shekfeh, Elisabeth-Maria Bissinger, et al.Bioorganic & Medicinal Chemistry|January 29, 2011
Lipophilic derivatives of leu-enkephalinamide: in vitro permeability, stability and in vivo nasal deliveryCécile D Cros, Istvan Toth, Joanne T BlanchfieldBioorganic & Medicinal Chemistry|January 11, 2011
Amyrin esters induce cell death by apoptosis in HL-60 leukemia cellsFrancisco W A Barros, Paulo N Bandeira, Daisy J B Lima, et al.Pageof 1,701