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Bioorganic & Medicinal Chemistry Letters|May 8, 2018
Discovery and optimization of aspartate aminotransferase 1 inhibitors to target redox balance in pancreatic ductal adenocarcinomaJustin Anglin, Reza Beheshti Zavareh, Philipp N Sander, et al.Bioorganic & Medicinal Chemistry Letters|May 8, 2018
Covalent inhibitors of nicotinamide N-methyltransferase (NNMT) provide evidence for target engagement challenges in situHsin-Yu Lee, Radu M Suciu, Benjamin D Horning, et al.Bioorganic & Medicinal Chemistry Letters|April 5, 2018
Benzoxazine derivatives of phytophenols show anti-plasmodial activity via sodium homeostasis disruptionVijeta Sharma, Nagarjuna Amarnath, Swapnil Shukla, et al.Bioorganic & Medicinal Chemistry Letters|April 5, 2018
A review of salvinorin analogs and their kappa-opioid receptor activityJeremy J Roach, Ryan A ShenviBioorganic & Medicinal Chemistry Letters|April 5, 2018
Synthesis of alkyne-tagged and biotin-tagged Sortin1 as novel photoaffinity probesRina Komatsu, Tamayo Yamaguchi, Naohiro Kobayashi, et al.Bioorganic & Medicinal Chemistry Letters|April 9, 2018
Design, synthesis and biological evaluation of seco-A-pentacyclic triterpenoids-3,4-lactone as potent non-nucleoside HBV inhibitorsZhijian Li, Qingxi Min, Haoji Huang, et al.Bioorganic & Medicinal Chemistry Letters|April 10, 2018
Novel thioureido-benzenesulfonamide derivatives with enaminone linker as potent anticancer, radiosensitizers and VEGFR2 inhibitorsMostafa M Ghorab, Fatma A Ragab, Helmy I Heiba, et al.Bioorganic & Medicinal Chemistry Letters|April 21, 2018
Synthesis and evaluation of new 2-chloro-4-aminopyrimidine and 2,6-dimethyl-4-aminopyrimidine derivatives as tubulin polymerization inhibitorsShaoyu Xu, Baijiao An, Yuxin Li, et al.Bioorganic & Medicinal Chemistry Letters|April 21, 2018
Synthesis of some novel dimethine, bis-dimethine cyanine dyes and octacosamethine cyanine dyes endowed with promising biological potency against (HepG2), (Hela), (MCF-7), (MIA), (SN12C) and (H358) cell linesRasha E El-Mekawy, A A FaddaBioorganic & Medicinal Chemistry Letters|April 26, 2018
Development of piperazine-based hydroxamic acid inhibitors against falcilysin, an essential malarial proteaseJeffrey P Chance, Hannah Fejzic, Obiel Hernandez, et al.Pageof 2,632