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Bioorganic & Medicinal Chemistry Letters|May 30, 2018
Synthesis of C-ring-modified blebbistatin derivatives and evaluation of their myosin II ATPase inhibitory potencyBart I Roman, Sigrid Verhasselt, Christophe W Mangodt, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2018
Discovery of chiral dihydropyridopyrimidinones as potent, selective and orally bioavailable inhibitors of AKTSaravanan Parthasarathy, Kenneth Henry, Huaxing Pei, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2018
Modular synthesis of new C-aryl-nucleosides and their anti-CML activityHamid Marzag, Marwa Zerhouni, Hamza Tachallait, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2018
Polyprenylated polycyclic acylphloroglucinol: Angiogenesis inhibitor from Garcinia multifloraLin-Yang Cheng, Chun-Lin Chen, Yueh-Hsiung Kuo, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2018
Catalytic asymmetric synthesis of α-methyl-p-boronophenylalanineShingo Harada, Ryota Kajihara, Risa Muramoto, et al.Bioorganic & Medicinal Chemistry Letters|April 15, 2018
An orally available, brain-penetrant CAMKK2 inhibitor reduces food intake in rodent modelDaniel J Price, David H Drewry, Lee T Schaller, et al.Bioorganic & Medicinal Chemistry Letters|August 29, 2016
Imaging human melanoma using a novel Tc-99m-labeled lactam bridge-cyclized alpha-MSH peptideLiqin Liu, Jingli Xu, Jianquan Yang, et al.Bioorganic & Medicinal Chemistry Letters|August 29, 2016
Indole-based allosteric inhibitors of HIV-1 integrasePratiq A Patel, Nina Kvaratskhelia, Yara Mansour, et al.Bioorganic & Medicinal Chemistry Letters|August 30, 2016
Bioactive diterpenoids from Trigonostemon chinensis: Structures, NO inhibitory activities, and interactions with iNOSJing Xu, Maoqin Peng, Xiaocong Sun, et al.Bioorganic & Medicinal Chemistry Letters|August 31, 2016
Pharbilignan C induces apoptosis through a mitochondria-mediated intrinsic pathway in human breast cancer cellsYong Joo Park, Chang-Ik Choi, Kyu Hyuck Chung, et al.Pageof 2,632