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Bioorganic & Medicinal Chemistry Letters|March 28, 2016
Dioxol and dihydrodioxin analogs of 2- and 3-phenylacetonitriles as potent anti-cancer agents with nanomolar activity against a variety of human cancer cellsNikhil R Madadi, Amit Ketkar, Narsimha R Penthala, et al.Bioorganic & Medicinal Chemistry Letters|March 30, 2016
An evaluation of synthetic indole derivatives as inhibitors of monoamine oxidaseZhanna V Chirkova, Mariya V Kabanova, Sergey I Filimonov, et al.Bioorganic & Medicinal Chemistry Letters|April 2, 2016
L-Aspartic and l-glutamic acid ester-based ProTides of anticancer nucleosides: Synthesis and antitumoral evaluationLing-Jie Gao, Steven De Jonghe, Dirk Daelemans, et al.Bioorganic & Medicinal Chemistry Letters|April 2, 2016
Development and evaluation of a highly reliable assay for SUMO-specific protease inhibitorsWenjuan Xie, Zhongli Wang, Jianchen Zhang, et al.Bioorganic & Medicinal Chemistry Letters|April 3, 2016
Strigolactone derivatives for potential crop enhancement applicationsClaudio Screpanti, Raymonde Fonné-Pfister, Alexandre Lumbroso, et al.Bioorganic & Medicinal Chemistry Letters|March 25, 2016
Paecilonic acids A and B, bicyclic fatty acids from the jellyfish-derived fungus Paecilomyces variotii J08NF-1Haibo Wang, Jongki Hong, Jun Yin, et al.Bioorganic & Medicinal Chemistry Letters|February 10, 2016
Synthesis and radiolabeling of (64)Cu-labeled 2-nitroimidazole derivative (64)Cu-BMS2P2 for hypoxia imagingZheng Luo, Hua Zhu, Xinfeng Lin, et al.Bioorganic & Medicinal Chemistry Letters|February 10, 2016
Carbonic anhydrase activators: Activation of the β-carbonic anhydrase from Malassezia globosa with amines and amino acidsDaniela Vullo, Sonia Del Prete, Clemente Capasso, et al.Bioorganic & Medicinal Chemistry Letters|February 13, 2016
In silico to in vitro screening of hydroxypyridinones as acetylcholinesterase inhibitorsMaria A Telpoukhovskaia, Brian O Patrick, Cristina Rodríguez-Rodríguez, et al.Bioorganic & Medicinal Chemistry Letters|May 11, 2016
Discovery of novel non-steroidal reverse indole mineralocorticoid receptor antagonistsAnthony K Ogawa, Ellen Vande Bunte, Rudrajit Mal, et al.Pageof 2,631