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Bioorganic & Medicinal Chemistry Letters|April 16, 2016
Discovery of biaryls as RORγ inverse agonists by using structure-based designIstvan J Enyedy, Noel A Powell, Justin Caravella, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2016
Structure-activity relationship study of 4-substituted piperidines at Leu26 moiety of novel p53-hDM2 inhibitorsYuan Tian, Yao Ma, Craig R Gibeau, et al.Bioorganic & Medicinal Chemistry Letters|April 16, 2016
Novel pyrazole derivatives with oxa/thiadiazolyl, pyrazolyl moieties and pyrazolo[4,3-d]-pyrimidine derivatives as potential antimicrobial and anticancer agentsHend N Hafez, Abdel-Rhman B A El-Gazzar, Sami A Al-HussainBioorganic & Medicinal Chemistry Letters|February 15, 2016
Synthesis of linear and cyclic peptide-PEG-lipids for stabilization and targeting of cationic liposome-DNA complexesKai K Ewert, Venkata Ramana Kotamraju, Ramsey N Majzoub, et al.Bioorganic & Medicinal Chemistry Letters|February 15, 2016
Synthesis and anticancer evaluation of spermatinamine analoguesBasem A Moosa, Sunil Sagar, Song Li, et al.Bioorganic & Medicinal Chemistry Letters|February 16, 2016
Novel indole sulfides as potent HIV-1 NNRTIsSiobhan Brigg, Nicole Pribut, Adriaan E Basson, et al.Bioorganic & Medicinal Chemistry Letters|February 16, 2016
Synthesis and anti-inflammatory activity evaluation of a novel series of 6-phenoxy-[1,2,4]triazolo[3,4-a]phthalazine-3-carboxamide derivativesDa-Chuan Liu, Guo-Hua Gong, Cheng-Xi Wei, et al.Bioorganic & Medicinal Chemistry Letters|February 26, 2016
Synthesis and preliminary evaluation of 5,7-dimethyl-2-aryl-3H-pyrrolizin-3-ones as angiogenesis inhibitorsNicholas S Kirk, Anna Bezos, Anthony C Willis, et al.Bioorganic & Medicinal Chemistry Letters|February 26, 2016
Synthesis, biological evaluation and molecular docking studies of 2-piperazin-1-yl-quinazolines as platelet aggregation inhibitors and ligands of integrin αIIbβ3Andrei A Krysko, Alexander Yu Kornylov, Pavel G Polishchuk, et al.Bioorganic & Medicinal Chemistry Letters|February 27, 2016
Anticancer activity studies of cubebin isolated from Piper cubeba and its synthetic derivativesDhanya S Rajalekshmi, Farha A Kabeer, Arya R Madhusoodhanan, et al.Pageof 2,631