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Bioorganic & Medicinal Chemistry Letters|April 7, 2020
Identification of a new class of non-electrophilic TRPA1 agonists by a structure-based virtual screening approachMitsugu Araki, Naoto Kanda, Hiroaki Iwata, et al.Bioorganic & Medicinal Chemistry Letters|August 28, 2020
Structure activity relationship exploration of 5-hydroxy-2-(3-phenylpropyl)chromones as a unique 5-HT2B receptor antagonist scaffoldMinsoo Kim, Myles Truss, Piyusha P Pagare, et al.Bioorganic & Medicinal Chemistry Letters|August 28, 2020
Design, synthesis and biological evaluation of triaryl compounds as novel 20S proteasome inhibitorsYajun Yang, Ke Wang, Bo Wu, et al.Bioorganic & Medicinal Chemistry Letters|August 28, 2020
Methods to optimize CNS exposure of drug candidatesNandini C PatelBioorganic & Medicinal Chemistry Letters|October 2, 2020
A carboxylic acid isostere screen of the DHODH inhibitor BrequinarLindsey G DeRatt, E Christine Pietsch, Alexandra Tanner, et al.Bioorganic & Medicinal Chemistry Letters|October 3, 2020
Reactive Pt(II) center as part of redox-active quinoline-based heterocyclic scaffolds toward new anticancer leadsSateeshkumar Kumbhakonam, Soumya Saroj, Nalini Venkatesan, et al.Bioorganic & Medicinal Chemistry Letters|March 10, 2020
Antibacterial activity of singly and doubly modified salinomycin derivativesMichał Sulik, Karolina Stępień, Joanna Stefańska, et al.Bioorganic & Medicinal Chemistry Letters|March 11, 2020
Synthesis and in vitro evaluation of antimycobacterial and cytotoxic activity of new α,β-unsaturated amide, oxazoline and oxazole derivatives from l-serineSaúl A Aguirre-Rentería, Juan J J Carrizales-Castillo, María Del Rayo Camacho Corona, et al.Bioorganic & Medicinal Chemistry Letters|March 23, 2020
Simplistic perylene-related compounds as inhibitors of tick-borne encephalitis virus reproductionNikita A Slesarchuk, Evgeny V Khvatov, Alexey A Chistov, et al.Bioorganic & Medicinal Chemistry Letters|March 18, 2020
Synthesis and pharmacokinetic study of a 11C-labeled cholesterol 24-hydroxylase inhibitor using 'in-loop' [11C]CO2 fixation methodZhen Chen, Jiahui Chen, Natalia Mast, et al.Pageof 2,631