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Bioorganic & Medicinal Chemistry Letters|November 1, 2023
Direct evaluation of polarity of the ligand binding pocket in retinoid X receptor using a fluorescent solvatochromic agonistKizuku Miura, Michiko Fujihara, Masaki Watanabe, et al.Bioorganic & Medicinal Chemistry Letters|November 18, 2023
Design, synthesis and antitubercular assessment of 1, 2, 3-triazole incorporated thiazolylcarboxylate derivativesRajubai D Bakale, Shubham M Sulakhe, Sanghratna L Kasare, et al.Bioorganic & Medicinal Chemistry Letters|November 15, 2023
Novel amino- and hydroxy-functionalized 1,2,4-trioxanes and their antimalarial activity against multidrug-resistant Plasmodium yoelii nigeriensis in Swiss mice via intramuscular and oral routePriyanka Yadav, Niraj Krishna Naikade, Mohammad Hassam, et al.Bioorganic & Medicinal Chemistry Letters|November 10, 2023
Discovery of (S)-3-(4-(benzyloxy)phenyl)-2-(2-phenoxyacetamido)propanoic acid derivatives as a new class of GPR34 antagonistsPei Zhou, Jinlong Zhao, Qian Hu, et al.Bioorganic & Medicinal Chemistry Letters|November 8, 2023
Discovery of a novel tetrahydroimidazo[1,2-a]pyridine-5-carboxylic acid derivative as a potent and selective heparanase-1 inhibitor utilizing an improved synthetic approachYudai Imai, Ryo Suzuki, Daisuke Matsuda, et al.Bioorganic & Medicinal Chemistry Letters|September 13, 2023
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamidesSuleyman Akocak, Nebih Lolak, Simone Giovannuzzi, et al.Bioorganic & Medicinal Chemistry Letters|September 9, 2023
Design, synthesis, and biological evaluation of THIQ as antidepressive agentsXiaopeng Wei, Man Zhang, Yijing Guo, et al.Bioorganic & Medicinal Chemistry Letters|August 9, 2023
Polyheterocyclic peptidomimetics: Parallel solid phase synthesis of oligo cyclic guanidines and their inhibition activity against Mycobacterium tuberculosis DNA gyraseMukund Tantak, Ramanjaneyulu Rayala, Zifang Deng, et al.Bioorganic & Medicinal Chemistry Letters|August 9, 2023
Short synthesis of a broadly Reactive, cell permeable serine hydrolase Fluorophosphonate-Alkyne probeSrihari Konduri, Joshua Schweer, Dionicio SiegelBioorganic & Medicinal Chemistry Letters|August 11, 2023
Enzymatic reconstitution of salicylate formation in promysalin biosynthesisSimita Das, Krushnamurthy Pattanayakanahalli Henjarappa, Nilkamal MahantaPageof 2,631