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Bioorganic & Medicinal Chemistry Letters|October 27, 2015
Synthesis and evaluation of antibacterial activity of (R)-2-methylheptyl isonicotinate, a putative naturally occurring bioactive agentJia Cao, Ben Adler, Patrick PerlmutterBioorganic & Medicinal Chemistry Letters|October 29, 2015
Discovery of an orally bioavailable isoxazoline benzoxaborole (AN8030) as a long acting animal ectoparasiticideYong-Kang Zhang, Jacob J Plattner, Eric E Easom, et al.Bioorganic & Medicinal Chemistry Letters|November 7, 2015
Synthesis, biological activity evaluation and molecular docking studies of novel coumarin substituted thiazolyl-3-aryl-pyrazole-4-carbaldehydesKrishnaiah Vaarla, Rajesh Kumar Kesharwani, Karnewar Santosh, et al.Bioorganic & Medicinal Chemistry Letters|November 8, 2015
PPL catalyzed four-component PASE synthesis of 5-monosubstituted barbiturates: Structure and pharmacological propertiesManisha Bihani, Pranjal P Bora, Alakesh K Verma, et al.Bioorganic & Medicinal Chemistry Letters|November 8, 2015
Discovery of novel 2-benzylisoquinolin-1(2H)-ones as potent vasodilative agentsBo-Rui Kang, Sen Li, Shuai Mao, et al.Bioorganic & Medicinal Chemistry Letters|November 9, 2015
Design and synthesis of an in vivo-efficacious PIM3 kinase inhibitor as a candidate anti-pancreatic cancer agentHirofumi Nakano, Tsukasa Hasegawa, Nae Saito, et al.Bioorganic & Medicinal Chemistry Letters|November 4, 2015
An abietane diterpene from Salvia cuspidata and some new derivatives are active against Trypanosoma cruziE S Lozano, R M Spina, C E Tonn, et al.Bioorganic & Medicinal Chemistry Letters|November 4, 2015
Solid-supported reagents composed of a copolymer possessing 2-O-sulfonyl mannosides and phase-transfer catalysts for the synthesis of 2-fluoroglucoseRyota Takeuchi, Yuki Sakai, Hiroshi Tanaka, et al.Bioorganic & Medicinal Chemistry Letters|November 4, 2015
A selective delta opioid receptor antagonist based on a stilbene coreAlyssa M Hartung, Hernan A Navarro, David F Wiemer, et al.Bioorganic & Medicinal Chemistry Letters|November 4, 2015
A novel class of negative allosteric modulators of NMDA receptor functionBrooke M Katzman, Riley E Perszyk, Hongjie Yuan, et al.Pageof 2,631