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Bioorganic & Medicinal Chemistry Letters|September 5, 2020
Structure-based amelioration of PXR transactivation in a novel series of macrocyclic allosteric inhibitors of HIV-1 integrasePrasanna Sivaprakasam, Zhongyu Wang, Nicholas A Meanwell, et al.Bioorganic & Medicinal Chemistry Letters|September 5, 2020
Synthesis of functionalized derivatives of the gamma-secretase modulator BMS-932481 and identification of its major metaboliteYunhui Zhang, Kenneth M Boy, Yong-Jin Wu, et al.Bioorganic & Medicinal Chemistry Letters|September 21, 2020
Discovery of a series of ester-substituted NLRP3 inflammasome inhibitorsDavid Harrison, Nicolas Boutard, Krzysztof Brzozka, et al.Bioorganic & Medicinal Chemistry Letters|September 8, 2020
Fragment-based lead discovery of a novel class of small molecule antagonists of neuropeptide B/W receptor subtype 1 (GPR7)Remond Moningka, F Anthony Romero, Nicholas B Hastings, et al.Bioorganic & Medicinal Chemistry Letters|September 8, 2020
Probing the B- & C-rings of the antimalarial tetrahydro-β-carboline MMV008138 for steric and conformational constraintsSha Ding, Maryam Ghavami, Joshua H Butler, et al.Bioorganic & Medicinal Chemistry Letters|September 14, 2020
Biochemical, cellular and structural characterization of novel and selective ERK3 inhibitorsUlrich Grädler, Michael Busch, Birgitta Leuthner, et al.Bioorganic & Medicinal Chemistry Letters|September 14, 2020
Synthesis of metronidazole based thiazolidinone analogs as promising antiamoebic agentsMohammad Fawad Ansari, Afreen Inam, Kamal Ahmad, et al.Bioorganic & Medicinal Chemistry Letters|September 17, 2020
3-(Cyclopropylmethyl)-7-((4-(4-[11C]methoxyphenyl)piperidin-1-yl)methyl)-8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine: Synthesis and preliminary evaluation for PET imaging of metabotropic glutamate receptor subtype 2Katsushi Kumata, Yiding Zhang, Masanao Ogawa, et al.Bioorganic & Medicinal Chemistry Letters|September 25, 2020
Synthesis and pharmacological evaluation of 11-(1,6-dimethyl-1,2,3,6-tetrahydropyridin-4-yl)-5H-dibenzo[b,e][1,4]diazepines with clozapine-like receptor occupancy at dopamine D1/D2 receptorHitoshi Watanabe, Kyoji Ishida, Masanori Yamamoto, et al.Bioorganic & Medicinal Chemistry Letters|September 26, 2020
A guanidinium-based inhibitor of a type I isopentenyl diphosphate isomeraseWalid M Abdelmagid, Niusha Mahmoodi, Martin E TannerPageof 2,632